SCHEMBL6508756

SCHEMBL6508756

COc1ccc(C(O)(Cc2ccncc2)c2ccccc2)cc1C1OCCCO1

nearest known ligand 0.39

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
HTT P42858 1/20 0.39
SMN1; SMN2 Q16637 1/20 0.39
MEN1 O00255 1/20 0.37
KMT2A Q03164 1/20 0.37
CYP1A2 P05177 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37
HIF1A Q16665 1/20 0.37
KCNA5 P22460 1/20 0.37
PDE4A P27815 9/20 0.36
PDE4D Q08499 3/20 0.36
PDE4B Q07343 2/20 0.36
PDE4C Q08493 2/20 0.36
SLC6A2 P23975 4/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7672093 0.80 CYP1A2 (0.34) HTTSMN1; SMN2CYP1A2CYP3A4CYP2C9
SCHEMBL6508090 0.78 PDE4A (0.58) PDE4APDE4DPDE4BPDE4C
SCHEMBL7672088 0.74 CYP3A4 (0.39) SMN1; SMN2KMT2ACYP1A2CYP3A4CYP2C9
SCHEMBL7314363 0.72 PDE4A (0.54) PDE4APDE4DPDE4BPDE4C
SCHEMBL10896574 0.71 CYP2C9 (0.66) SMN1; SMN2MEN1KMT2ACYP1A2CYP3A4
SCHEMBL7900925 0.69 PDE4A (0.59) PDE4APDE4DPDE4BPDE4C
SCHEMBL7907983 0.69 PDE4A (0.50) PDE4APDE4DPDE4BPDE4C
SCHEMBL7911130 0.69 PDE4A (0.59) PDE4APDE4DPDE4BPDE4C
SCHEMBL6886593 0.69 PDE4A (0.51) PDE4APDE4DPDE4BPDE4C
SCHEMBL7138058 0.68 CYP2C19 (0.38) CYP2C19SLC6A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0766669-B1 TRI-SUBSTITUTED PHENYL DERIVATIVES USEFUL AS PDE IV INHIBITORS CELLTECH R&D LTD (GB) 2005-04-20 EP disclosed
US-6245774-B1 ANTIINFLAMMATORY AGENTS; BRONCHODILATOR AGENTS CELLTECH THERAPEUTICS LIMITED (GB) 2001-06-12 US disclosed