SCHEMBL6508768

SCHEMBL6508768

COc1cc(-c2ccoc2)nc(C(=O)O)c1O

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERN1 O75460 1/20 0.49
ATR Q13535 1/20 0.45
ADORA2A P29274 3/20 0.43
ADORA3 P0DMS8 2/20 0.43
ADORA2B P29275 2/20 0.43
PDGFRB P09619 1/20 0.43
FYN P06241 1/20 0.41
ADORA1 P30542 2/20 0.41
CA12 O43570 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
CA3 P07451 1/20 0.40
PKM P14618 1/20 0.40
CA4 P22748 1/20 0.40
CA6 P23280 1/20 0.40
CA5A P35218 1/20 0.40
CA7 P43166 1/20 0.40
CA9 Q16790 1/20 0.40
CA14 Q9ULX7 1/20 0.40
CA5B Q9Y2D0 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6371584 0.77 POLB (0.49) ATRALDH1A1MAPK1LMNAKMT2A
SCHEMBL17416879 0.72 PKM (0.50) ERN1FYNCA12CA1CA2
SCHEMBL19283132 0.69 PKM (0.50) ERN1FYNCA12CA1CA2
SCHEMBL19350459 0.68 CCR6 (0.51) ERN1ALDH1A1MAPK1LMNACYP1A2
SCHEMBL3586846 0.67 ATR (0.57) ATRMAPK1PLAUCYP3A4
SCHEMBL12767028 0.66 ERN1 (1.00) ERN1
SCHEMBL753212 0.66 CA12 (0.44) CA12CA1CA2CA3PKM
Hydrochloric Acid SCHEMBL5583653 0.64 CA12 (0.43) CA12CA1CA2CA3PKM
SCHEMBL6373026 0.64 MAPK1 (0.40) CA12CA1CA2CA3PKM
SCHEMBL26685065 0.64 PDGFRB (0.43) ADORA2AADORA3ADORA2BPDGFRBADORA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005042524-A1 PYRIDINE CARBOXAMIDE AND METHODS FOR INHIBITING HIV INTEGRASE VIROCHEM PHARMA INC. (CA) 2005-05-12 WO claimed
WO-2005042524-A1 PYRIDINE CARBOXAMIDE AND METHODS FOR INHIBITING HIV INTEGRASE VIROCHEM PHARMA INC. (CA) 2005-05-12 WO disclosed