SCHEMBL6508989

SCHEMBL6508989

COCCCN1C(=O)COc2ccc(I)cc21

nearest known ligand 0.56

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
REN P00797 1/20 0.56
TSHR P16473 3/20 0.55
KDM4E B2RXH2 1/20 0.47
POLB P06746 4/20 0.46
TP53 P04637 2/20 0.46
THRB P10828 2/20 0.46
MAPT P10636 1/20 0.46
KMO O15229 1/20 0.44
HTT P42858 1/20 0.43
DRD2 P14416 1/20 0.43
HTR2A P28223 1/20 0.43
MCHR1 Q99705 1/20 0.43
BRD4 O60885 1/20 0.43
KMT2A Q03164 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL89401 0.86 TSHR (0.71) RENTSHRPOLBTP53THRB
SCHEMBL1047741 0.86 REN (0.57) RENTSHRKDM4EPOLBTP53
SCHEMBL55503 0.85 REN (0.61) RENTSHRKDM4EPOLBTP53
SCHEMBL6721804 0.85 REN (0.56) RENTSHRKDM4EPOLBTP53
SCHEMBL3065160 0.84 REN (0.55) RENTSHRKDM4EPOLBTP53
SCHEMBL927855 0.84 REN (0.55) RENTSHRKDM4EPOLBTP53
SCHEMBL1015445 0.83 TSHR (0.56) RENTSHRKDM4EPOLBTP53
SCHEMBL8306331 0.83 REN (0.56) RENTSHRKDM4EPOLBTP53
SCHEMBL78468 0.83 REN (0.54) RENTSHRKDM4EPOLBTP53
SCHEMBL2339596 0.83 TSHR (0.56) RENTSHRKDM4EPOLBTP53

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1833816-B1 SUBSTITUTED PIPERIDINES AS RENIN INHIBITORS NOVARTIS AG (CH) 2009-11-11 EP disclosed
WO-2005037803-A1 ORGANIC COMPOUNDS SPEEDEL EXPERIMENTA AG (CH) 2005-04-28 WO disclosed