SCHEMBL6509749

SCHEMBL6509749

Cc1c(-c2ccccc2)nc2ncccc2c1C(=O)O

nearest known ligand 0.94

Predicted protein targets (top 3)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 17/20 0.94
PDE10A Q9Y233 3/20 0.68
TSHR P16473 1/20 0.68

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6509265 0.86 DHODH (0.72) DHODHPDE10ATSHR
SCHEMBL20659638 0.83 DHODH (0.68) DHODHPDE10ATSHR
SCHEMBL1581468 0.81 PDE10A (1.00) DHODHPDE10ATSHR
SCHEMBL9954367 0.80 DHODH (0.63) DHODHPDE10ATSHR
Hydrochloric Acid SCHEMBL27511204 0.80 PDE10A (0.97) DHODHPDE10ATSHR
SCHEMBL2124987 0.79 DHODH (0.62) DHODHPDE10ATSHR
SCHEMBL28170815 0.77 DHODH (0.73) DHODHPDE10ATSHR
SCHEMBL2807617 0.76 PDE10A (0.77) DHODHPDE10ATSHR
SCHEMBL18075791 0.75 PDE10A (0.75) DHODHPDE10ATSHR
SCHEMBL4228780 0.74 DHODH (0.70) DHODHPDE10ATSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005000845-A2 BICYCLIC DERIVATIVES AS NK-1 AND NK-2 ANTAGONISTS NIKEM RESEARCH S.R.L. (IT) 2005-01-06 WO disclosed