SCHEMBL6509265

SCHEMBL6509265

COC(=O)c1c(C)c(-c2ccccc2)nc2ncccc12

nearest known ligand 0.72

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 9/20 0.72
TSHR P16473 1/20 0.51
PDE10A Q9Y233 1/20 0.51
SMN1; SMN2 Q16637 1/20 0.50
TACR3 P29371 1/20 0.49
MEN1 O00255 1/20 0.46
KMT2A Q03164 1/20 0.46
PTGS1 P23219 1/20 0.46
MAPT P10636 1/20 0.46
GABRA1 P14867 2/20 0.45
GABRG2 P18507 2/20 0.45
GABRB3 P28472 2/20 0.45
GABRA5 P31644 2/20 0.45
GABRA3 P34903 2/20 0.45
ALDH1A1 P00352 1/20 0.45
GABRP O00591 1/20 0.44
GABRD O14764 1/20 0.44
GABRB1 P18505 1/20 0.44
GABRA2 P47869 1/20 0.44
GABRB2 P47870 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6509749 0.86 DHODH (0.94) DHODHTSHRPDE10A
SCHEMBL6506852 0.85 DHODH (0.56) DHODHTSHRPDE10ASMN1; SMN2TACR3
SCHEMBL2372674 0.83 PDE10A (0.73) DHODHTSHRPDE10ASMN1; SMN2TACR3
SCHEMBL9954367 0.76 DHODH (0.63) DHODHTSHRPDE10AMEN1KMT2A
SCHEMBL2459661 0.75 DHODH (0.72) DHODH
SCHEMBL2124987 0.75 DHODH (0.62) DHODHTSHRPDE10AMEN1KMT2A
SCHEMBL17594221 0.74 DHODH (0.71) DHODHTSHRPDE10A
SCHEMBL14553152 0.74 DHODH (0.95) DHODHPDE10A
SCHEMBL30690105 0.74 PLA2G2A (0.58) DHODHTSHRPDE10ATACR3MEN1
SCHEMBL5945348 0.73 DHODH (0.63) DHODHTSHRPDE10ASMN1; SMN2TACR3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005000845-A2 BICYCLIC DERIVATIVES AS NK-1 AND NK-2 ANTAGONISTS NIKEM RESEARCH S.R.L. (IT) 2005-01-06 WO disclosed