SCHEMBL6509894

SCHEMBL6509894

N#Cc1ccc(N(CCO)CCO)c(C(F)(F)F)c1

nearest known ligand 0.43

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
TRPV4 Q9HBA0 2/20 0.43
KIF11 P52732 2/20 0.39
MRGPRX4 Q96LA9 1/20 0.38
AR P10275 6/20 0.37
CYP19A1 P11511 2/20 0.37
SCN9A Q15858 3/20 0.35
P4HB P07237 1/20 0.35
TMPRSS4 Q9NRS4 1/20 0.34
ABCB1 P08183 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3410649 0.92 AR (0.44) TRPV4KIF11MRGPRX4ARCYP19A1
SCHEMBL3055456 0.84 TRPV4 (0.38) TRPV4KIF11MRGPRX4ARCYP19A1
SCHEMBL3527583 0.81 TRPV4 (0.45) TRPV4KIF11MRGPRX4ARCYP19A1
SCHEMBL11799852 0.78 GAA (0.38) ABCB1
SCHEMBL2584317 0.77 MRGPRX4 (0.44) TRPV4KIF11MRGPRX4ARCYP19A1
SCHEMBL3525556 0.76 TRPV4 (0.43) TRPV4KIF11MRGPRX4ARCYP19A1
SCHEMBL250976 0.76 TRPV4 (0.49) TRPV4KIF11MRGPRX4ARCYP19A1
SCHEMBL11804570 0.74 GAA (0.38) ABCB1
SCHEMBL6511318 0.73 SRD5A2 (0.42) MRGPRX4ARP4HB
SCHEMBL3051276 0.72 TRPV4 (0.40) TRPV4KIF11MRGPRX4ARCYP19A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6852755-B1 Nitrogen mustard compounds and prodrugs therefor CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2005-02-08 US disclosed
EP-1165493-B1 NITROGEN MUSTARD COMPOUNDS AND PRODRUGS THEREFOR CANCER REC TECH LTD (GB) 2005-01-19 EP disclosed
EP-1165493-A1 NITROGEN MUSTARD COMPOUNDS AND PRODRUGS THEREFOR CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2002-01-02 EP disclosed
WO-2000058271-A1 NITROGEN MUSTARD COMPOUNDS AND PRODRUGS THEREFOR CANCER RESEARCH CAMPAIGN TECHNOLOGY LIMITED (GB) 2000-10-05 WO disclosed