SCHEMBL6509987

SCHEMBL6509987

COc1ccc(CN2CCc3c(C(=O)N(C)C)nc(O)c(OC)c3C2=O)cc1.COc1ccc(CN2CCc3c(C(=O)N(C)C)nc(OC(C)=O)c(OC)c3C2=O)cc1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
GAA P10253 1/20 0.36
ALDH1A1 P00352 3/20 0.36
SMN1; SMN2 Q16637 2/20 0.36
CYP1A2 P05177 1/20 0.36
CYP2C19 P33261 1/20 0.36
KEAP1 Q14145 1/20 0.35
EGLN1 Q9GZT9 5/20 0.34
HDAC1 Q13547 2/20 0.34
HDAC3 O15379 1/20 0.34
HDAC4 P56524 1/20 0.34
HDAC7 Q8WUI4 1/20 0.34
HDAC2 Q92769 1/20 0.34
HDAC10 Q969S8 1/20 0.34
HDAC11 Q96DB2 1/20 0.34
HDAC8 Q9BY41 1/20 0.34
HDAC6 Q9UBN7 1/20 0.34
HDAC9 Q9UKV0 1/20 0.34
HDAC5 Q9UQL6 1/20 0.34
F2 P00734 2/20 0.34
F10 P00742 2/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4493594 0.96 GAA (0.39) GAAALDH1A1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL4490423 0.92 GAA (0.42) GAAALDH1A1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL6032330 0.86 KEAP1 (0.33) GAAALDH1A1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL4502970 0.75 EGLN1 (0.45) GAAALDH1A1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL5814580 0.75 TNIK (0.33) EGLN1
SCHEMBL4477518 0.73 GAA (0.42) GAAALDH1A1SMN1; SMN2CYP1A2CYP2C19
SCHEMBL4484200 0.73 LMNA (0.36) ALDH1A1SMN1; SMN2LMNAKMT2APOLB
SCHEMBL1335829 0.72 MEN1 (0.37) ALDH1A1SMN1; SMN2LMNAKMT2AMEN1
SCHEMBL4502946 0.71 AKR1B1 (0.43) ALDH1A1SMN1; SMN2EGLN1LMNAKMT2A
SCHEMBL5438443 0.70 GAA (0.42) GAAALDH1A1SMN1; SMN2CYP1A2CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005087767-A1 HIV INTEGRASE INHIBITORS MERCK & CO., INC. (US) 2005-09-22 WO disclosed