SCHEMBL6510199

SCHEMBL6510199

CN1CCC[C@H]1C(=O)Nc1cc(C(N)=O)c(NC(N)=O)s1

nearest known ligand 0.48

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP3A4 P08684 1/20 0.48
CYP2D6 P10635 1/20 0.48
IKBKB O14920 4/20 0.44
PARP1 P09874 2/20 0.43
CHEK1 O14757 7/20 0.43
MAPK1 P28482 1/20 0.42
GFER P55789 1/20 0.42
JAK2 O60674 2/20 0.40
MEN1 O00255 1/20 0.40
EIF2AK2 P19525 1/20 0.40
KMT2A Q03164 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
JAK3 P52333 1/20 0.39
USP2 O75604 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
HSD17B10 Q99714 2/20 0.38
MAPT P10636 1/20 0.38
ALOX15 P16050 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6510188 1.00 CYP3A4 (0.48) CYP3A4CYP2D6IKBKBPARP1CHEK1
SCHEMBL6509261 0.81 MAPK1 (0.49) IKBKBPARP1CHEK1MAPK1GFER
SCHEMBL6507196 0.74 MAPK1 (0.49) IKBKBCHEK1MAPK1GFERJAK2
SCHEMBL6530224 0.74 MAPK1 (0.49) IKBKBCHEK1MAPK1GFERJAK2
Hydrochloric Acid SCHEMBL6506232 0.73 MAPK1 (0.48) IKBKBCHEK1MAPK1GFERJAK2
SCHEMBL6509035 0.73 MAPK1 (0.48) IKBKBCHEK1MAPK1GFERJAK2
SCHEMBL6530184 0.72 CHEK1 (0.48) IKBKBCHEK1MAPK1GFER
SCHEMBL6507091 0.70 CHEK1 (0.47) IKBKBCHEK1MAPK1GFERMEN1
SCHEMBL6507207 0.70 MAPK1 (0.47) IKBKBCHEK1MAPK1GFERJAK2
SCHEMBL6511679 0.68 IKBKB (0.48) IKBKBCHEK1MAPK1GFERJAK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed