SCHEMBL6511017

SCHEMBL6511017

CCOc1ccc(-c2nnc(C)n2-c2ccc(OC)nc2)cc1Cl

nearest known ligand 0.80

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
OXTR P30559 19/20 0.80
AVPR1A P37288 9/20 0.78
AVPR2 P30518 3/20 0.59
TUBB4A P04350 1/20 0.47
TUBB P07437 1/20 0.47
TUBA3C P0DPH7 1/20 0.47
TUBA1B P68363 1/20 0.47
TUBA4A P68366 1/20 0.47
TUBB4B P68371 1/20 0.47
TUBB3 Q13509 1/20 0.47
TUBB2A Q13885 1/20 0.47
TUBB8 Q3ZCM7 1/20 0.47
TUBA3E Q6PEY2 1/20 0.47
TUBA1A Q71U36 1/20 0.47
TUBA1C Q9BQE3 1/20 0.47
TUBB6 Q9BUF5 1/20 0.47
TUBB2B Q9BVA1 1/20 0.47
TUBB1 Q9H4B7 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8282112 0.89 OXTR (1.00) OXTRAVPR1AAVPR2
SCHEMBL6510715 0.87 OXTR (0.87) OXTRAVPR1AAVPR2TUBB4ATUBB
SCHEMBL8282084 0.77 OXTR (0.81) OXTRAVPR1AAVPR2
SCHEMBL8281669 0.76 OXTR (0.77) OXTRAVPR1AAVPR2
SCHEMBL8281027 0.76 OXTR (1.00) OXTRAVPR1AAVPR2
SCHEMBL17367287 0.76 OXTR (0.69) OXTRAVPR1AAVPR2
SCHEMBL8280934 0.75 OXTR (0.81) OXTRAVPR1AAVPR2
SCHEMBL8279809 0.75 OXTR (0.68) OXTRAVPR1AAVPR2
SCHEMBL8282609 0.74 OXTR (1.00) OXTRAVPR1AAVPR2
SCHEMBL15840847 0.74 OXTR (0.60) OXTRAVPR1AAVPR2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed