SCHEMBL6511862

SCHEMBL6511862

FC(F)(F)c1cc(CCCCBr)cc(C(F)(F)F)c1

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 2/20 0.44
DAO P14920 2/20 0.41
TACR1 P25103 9/20 0.40
CES2 O00748 1/20 0.39
SIRT2 Q8IXJ6 1/20 0.37
TAAR1 Q96RJ0 1/20 0.36
HDAC1 Q13547 1/20 0.36
HDAC8 Q9BY41 1/20 0.36
MLYCD O95822 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL81976 0.94 IDO1 (0.45) IDO1DAOTACR1CES2SIRT2
SCHEMBL2393670 0.85 IDO1 (0.48) IDO1DAOTACR1CES2TAAR1
SCHEMBL7384474 0.80 TAAR1 (0.59) IDO1DAOTAAR1HDAC1HDAC8
SCHEMBL16298283 0.80 TAAR1 (0.59) IDO1DAOTAAR1HDAC1HDAC8
SCHEMBL5781780 0.79 TAAR1 (0.55) IDO1SIRT2TAAR1HDAC1HDAC8
SCHEMBL7574477 0.79 RAD52 (0.49) IDO1DAOTACR1TAAR1
SCHEMBL14402519 0.79 PTGS2 (0.50) IDO1DAOTACR1
SCHEMBL7777598 0.78 RAD52 (0.48) IDO1DAOTACR1TAAR1
SCHEMBL28703223 0.78 RAD52 (0.48) IDO1DAOTACR1TAAR1
SCHEMBL6231341 0.78 RAD52 (0.48) IDO1DAOTACR1TAAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005080354-A1 1,2,4-TRIAZINES DERIVATIVES, PREPARATION THEREOF AND USE THEREOF IN HUMAN THERAPEUTICS PIERRE FABRE MEDICAMENT (FR) 2005-09-01 WO disclosed