SCHEMBL6512302

SCHEMBL6512302

O=C(O)CC(NC(=O)/C=C/c1ccccc1)c1ccc(NC(=O)c2c(Cl)cncc2Cl)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
EGFR P00533 3/20 0.47
UTS2R Q9UKP6 2/20 0.47
ITGB1 P05556 5/20 0.47
ITGA4 P13612 5/20 0.47
MMP1 P03956 3/20 0.45
MMP2 P08253 3/20 0.45
MMP9 P14780 3/20 0.45
LMNA P02545 2/20 0.42
NPSR1 Q6W5P4 2/20 0.42
MEN1 O00255 2/20 0.42
MAPT P10636 2/20 0.42
KMT2A Q03164 2/20 0.42
CYP1A2 P05177 1/20 0.42
CYP3A4 P08684 1/20 0.42
CYP2D6 P10635 1/20 0.42
CYP2C9 P11712 1/20 0.42
CYP2C19 P33261 1/20 0.42
CTSA P10619 1/20 0.41
MAOA P21397 1/20 0.41
MAOB P27338 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6512308 1.00 EGFR (0.47) EGFRUTS2RITGB1ITGA4MMP1
SCHEMBL6509549 0.84 ITGB1 (0.63) ITGB1ITGA4CTSA
SCHEMBL6513196 0.80 ITGB1 (0.53) ITGB1ITGA4KMT2A
SCHEMBL6512395 0.79 ITGB1 (0.49) ITGB1ITGA4KMT2A
SCHEMBL6520177 0.78 ITGB1 (0.52) ITGB1ITGA4LMNANPSR1CTSA
SCHEMBL6509698 0.78 ITGB1 (0.48) ITGB1ITGA4RAB9A
SCHEMBL6512380 0.78 ITGA4 (0.50) ITGB1ITGA4
SCHEMBL6509525 0.77 ITGB1 (0.52) ITGB1ITGA4LMNAMEN1MAPT
SCHEMBL6514009 0.77 ITGB1 (0.58) ITGB1ITGA4MEN1MAPTKMT2A
SCHEMBL6518236 0.77 ITGB1 (0.52) ITGB1ITGA4LMNACTSARAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6953798-B1 β-alanine derivates CELLTECH R&D LIMITED (GB) 2005-10-11 US disclosed