SCHEMBL651425

SCHEMBL651425

CCCCn1c(-c2ccccc2)nc(-c2ccc(OC)cc2)c1CC(COC)NCc1ccc(C(N)=O)c(O)c1

nearest known ligand 0.35

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
MTNR1B P49286 1/20 0.35
ATM Q13315 3/20 0.35
PARP1 P09874 2/20 0.34
ALDH1A1 P00352 2/20 0.34
HPGD P15428 2/20 0.34
C5AR1 P21730 1/20 0.34
MEN1 O00255 1/20 0.34
KMT2A Q03164 1/20 0.34
BCHE P06276 3/20 0.33
GAA P10253 2/20 0.33
MAPT P10636 1/20 0.33
DHODH Q02127 1/20 0.33
ROCK2 O75116 1/20 0.33
CD38 P28907 1/20 0.33
IRAK4 Q9NWZ3 1/20 0.33
KDM4E B2RXH2 1/20 0.33
SMN1; SMN2 Q16637 1/20 0.33
HSD17B10 Q99714 1/20 0.33
PPARG P37231 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL648736 0.91 ATM (0.36) ATMPARP1ALDH1A1C5AR1MEN1
SCHEMBL651426 0.81 C5AR1 (0.38) PARP1ALDH1A1HPGDC5AR1MEN1
SCHEMBL648253 0.81 TSHR (0.41) PARP1C5AR1MAPTPPARG
SCHEMBL650278 0.81 C5AR1 (0.40) PARP1C5AR1PPARG
SCHEMBL648586 0.80 C5AR1 (0.39) PARP1C5AR1BCHEMAPTPPARG
SCHEMBL648873 0.79 MC4R (0.37) ATMPARP1C5AR1MEN1KMT2A
SCHEMBL649230 0.79 C5AR1 (0.38) PARP1ALDH1A1C5AR1MEN1KMT2A
SCHEMBL648105 0.76 C5AR1 (0.38) PARP1ALDH1A1C5AR1MEN1KMT2A
SCHEMBL648963 0.76 C5AR1 (0.54) ALDH1A1HPGDC5AR1MEN1KMT2A
SCHEMBL14572934 0.74 PDK1 (0.40) PARP1MAPTPPARG

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119665-B2 Aryl imidazoles and related compounds as C5a receptor modulators NOVARTIS INTERNATIONAL PHARMACEUTICAL LTD. (BM) 2012-02-21 US disclosed