SCHEMBL651516

SCHEMBL651516

CC(C)(C)N(C(=O)O)c1ccc(-c2ccsc2)cc1NC(=O)c1ccc(N)cc1

nearest known ligand 0.53

Predicted protein targets (top 7)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 15/20 0.53
HDAC2 Q92769 6/20 0.44
P2RY14 Q15391 1/20 0.41
HDAC3 O15379 4/20 0.40
CHEK2 O96017 1/20 0.40
KCNH2 Q12809 3/20 0.40
MAP3K5 Q99683 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL653154 0.84 HDAC1 (0.45) HDAC1HDAC2CHEK2KCNH2
SCHEMBL651416 0.84 HDAC1 (0.58) HDAC1HDAC2HDAC3KCNH2
SCHEMBL4120548 0.79 HDAC1 (0.76) HDAC1HDAC2HDAC3KCNH2
SCHEMBL653107 0.79 KCNH2 (0.49) HDAC1CHEK2KCNH2
SCHEMBL4126494 0.78 HDAC1 (0.58) HDAC1HDAC2P2RY14HDAC3CHEK2
SCHEMBL2684526 0.77 HDAC1 (0.45) HDAC1HDAC2P2RY14HDAC3
SCHEMBL4282116 0.76 HDAC1 (0.54) HDAC1HDAC2P2RY14HDAC3CHEK2
SCHEMBL1930616 0.75 HDAC1 (0.64) HDAC1HDAC2HDAC3
SCHEMBL1931248 0.73 HDAC1 (0.55) HDAC1HDAC2HDAC3
SCHEMBL1931108 0.73 HDAC1 (0.53) HDAC1HDAC2HDAC3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119685-B2 Disubstituted aniline compounds MERCK SHARP & DOHME CORP. (US) 2012-02-21 US disclosed