SCHEMBL6516516

SCHEMBL6516516

CCOc1cc(-c2c(CC)cccc2CC)ncc1CCCCOc1cccc(C(=O)OC)c1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
CYP1A2 P05177 1/20 0.41
CYP3A4 P08684 1/20 0.41
CYP2D6 P10635 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41
CYSLTR1 Q9Y271 1/20 0.41
SMPD1 P17405 3/20 0.40
KMT2A Q03164 2/20 0.40
CREBBP Q92793 1/20 0.38
MEN1 O00255 1/20 0.38
POLB P06746 1/20 0.38
MDH1 P40925 1/20 0.38
THRA P10827 1/20 0.38
THRB P10828 1/20 0.38
CYP4F2 P78329 1/20 0.38
CYP4A11 Q02928 1/20 0.38
MTNR1A P48039 1/20 0.37
MTNR1B P49286 1/20 0.37
NR1H4 Q96RI1 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6515014 0.83 MAPK1 (0.40) CYP2D6POLB
SCHEMBL1327155 0.81 CREBBP (0.38) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL6518505 0.79 C5AR1 (0.37) ALDH1A1CYP4F2CYP4A11
SCHEMBL6522088 0.78 NPSR1 (0.36) ALDH1A1POLBTHRB
SCHEMBL1327243 0.77 PPARG (0.47) ALDH1A1CYSLTR1KMT2ACREBBPPOLB
SCHEMBL6523352 0.75 C5AR1 (0.38)
SCHEMBL1327217 0.73 KMT2A (0.44) KMT2APOLBNR1H4
SCHEMBL7322482 0.72 SMPD1 (0.70) ALDH1A1CYP1A2CYP3A4CYP2D6CYP2C9
SCHEMBL644216 0.72 SMN1; SMN2 (0.58) ALDH1A1CYSLTR1KMT2AMEN1POLB
SCHEMBL31442462 0.72 SMN1; SMN2 (0.58) ALDH1A1CYSLTR1KMT2AMEN1POLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565452-A2 3-SUBSTITUTED-6-ARYL PYRIDINES AS LIGANDS OF C5A RECEPTORS NEUROGEN CORPORATION (US) 2005-08-24 EP disclosed
WO-2004043925-A2 3-SUBSTITUTED-6-ARYL PYRIDINED AS LIGANDS OF C5A RECEPTORS NEUROGEN CORPORATION (US) 2004-05-27 WO disclosed