SCHEMBL6522088

SCHEMBL6522088

CCOc1cc(-c2c(CC)cccc2CC)ncc1CCCCCl

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 2/20 0.36
MAPT P10636 2/20 0.36
L3MBTL1 Q9Y468 1/20 0.36
C5AR1 P21730 4/20 0.35
KDM4E B2RXH2 1/20 0.34
NPC1 O15118 1/20 0.34
MITF O75030 1/20 0.34
THRB P10828 1/20 0.34
MAPK1 P28482 1/20 0.34
RAB9A P51151 1/20 0.34
GLS O94925 2/20 0.34
ELANE P08246 2/20 0.33
LMNA P02545 1/20 0.32
HTT P42858 1/20 0.32
ALDH1A1 P00352 2/20 0.32
POLB P06746 1/20 0.32
PTGS2 P35354 1/20 0.31
SLC6A2 P23975 4/20 0.31
SLC6A4 P31645 4/20 0.31
SLC6A3 Q01959 4/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6518505 0.89 C5AR1 (0.37) NPSR1MAPTL3MBTL1C5AR1GLS
SCHEMBL6515324 0.85 MAPT (0.41) NPSR1MAPTL3MBTL1KDM4EMAPK1
SCHEMBL6522038 0.83 C5AR1 (0.33) NPSR1MAPTL3MBTL1C5AR1
SCHEMBL1328160 0.81 C5AR1 (0.41) NPSR1MAPTL3MBTL1C5AR1ELANE
SCHEMBL6515014 0.80 MAPK1 (0.40) L3MBTL1MAPK1POLB
SCHEMBL6522043 0.80 PPARA (0.49) ELANEPTGS2
SCHEMBL6523352 0.79 C5AR1 (0.38) L3MBTL1C5AR1PTGS2
SCHEMBL6520800 0.79 ALOX5 (0.43) C5AR1ELANEPTGS2
SCHEMBL6516516 0.78 ALDH1A1 (0.41) THRBALDH1A1POLB
SCHEMBL6522026 0.76 S1PR1 (0.41) C5AR1PTGS2SLC6A2SLC6A4SLC6A3

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1565452-A2 3-SUBSTITUTED-6-ARYL PYRIDINES AS LIGANDS OF C5A RECEPTORS NEUROGEN CORPORATION (US) 2005-08-24 EP disclosed
WO-2004043925-A2 3-SUBSTITUTED-6-ARYL PYRIDINED AS LIGANDS OF C5A RECEPTORS NEUROGEN CORPORATION (US) 2004-05-27 WO disclosed