SCHEMBL6518331

SCHEMBL6518331

COc1nc(NC2CCC(N)CC2)nc(OC)n1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPSR1 Q6W5P4 4/20 0.50
HTT P42858 4/20 0.50
SMN1; SMN2 Q16637 2/20 0.50
ALDH1A1 P00352 3/20 0.42
CDK7 P50613 2/20 0.41
CDK9 P50750 2/20 0.41
MAPT P10636 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
MAPK6 Q16659 1/20 0.41
TSHR P16473 3/20 0.40
LMNA P02545 2/20 0.40
ROCK2 O75116 1/20 0.40
ROCK1 Q13464 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
PIM1 P11309 1/20 0.39
TP53 P04637 2/20 0.38
ALOX15 P16050 1/20 0.38
PDGFRA P16234 3/20 0.37
CCNE1 P24864 3/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6509364 0.79 HTT (0.50) NPSR1HTTSMN1; SMN2ALDH1A1MAPT
Hydrochloric Acid SCHEMBL3770176 0.77 HTT (0.49) NPSR1HTTSMN1; SMN2ALDH1A1MAPT
SCHEMBL10964479 0.76 NPSR1 (0.51) NPSR1HTTSMN1; SMN2ALDH1A1MAPT
SCHEMBL10511471 0.75 NPSR1 (0.61) NPSR1HTTSMN1; SMN2ALDH1A1MAPT
SCHEMBL1412368 0.72 PDE4A (0.56) CDK7CDK9ROCK2ROCK1PIM1
SCHEMBL11274944 0.70 NPSR1 (0.45) NPSR1HTTSMN1; SMN2ALDH1A1MAPT
SCHEMBL6459225 0.70 CDK9 (0.49) CDK7CDK9MAPK6ROCK2ROCK1
SCHEMBL6459216 0.70 CDK9 (0.49) CDK7CDK9MAPK6ROCK2ROCK1
SCHEMBL10864593 0.70 ALDH1A1 (0.60) NPSR1HTTSMN1; SMN2ALDH1A1MAPT
SCHEMBL3774476 0.70 PDE4A (0.46) NPSR1HTTSMN1; SMN2ALDH1A1MAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005095339-A1 DICYANOPYRROLIDINES AS DIPEPTIDYL PEPTIDASE IV INHIBITORS PFIZER PRODUCTS INC. (US) 2005-10-13 WO disclosed