SCHEMBL6519271

SCHEMBL6519271

c1coc([C]2NCCN2)c1

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.52
ALDH1A1 P00352 6/20 0.44
KDM4E B2RXH2 5/20 0.44
MAPT P10636 4/20 0.44
POLB P06746 3/20 0.44
MEN1 O00255 3/20 0.44
KMT2A Q03164 3/20 0.44
HPGD P15428 3/20 0.44
BLM P54132 3/20 0.44
PKM P14618 3/20 0.44
HSD17B10 Q99714 3/20 0.44
TDP1 Q9NUW8 3/20 0.44
ALOX15 P16050 2/20 0.44
CASP1 P29466 2/20 0.44
PTPN7 P35236 2/20 0.44
RECQL P46063 2/20 0.44
CASP7 P55210 2/20 0.44
L3MBTL1 Q9Y468 2/20 0.44
RAB9A P51151 2/20 0.44
USP2 O75604 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1799678 0.73 ALDH1A1 (0.63) NISCHALDH1A1KDM4EMAPTPOLB
SCHEMBL6909709 0.70 NISCH (0.46) NISCHALDH1A1KDM4EMAPTPOLB
SCHEMBL1607474 0.69 NISCH (0.44) NISCHALDH1A1KDM4EMAPTPOLB
SCHEMBL498016 0.67
Piperazine SCHEMBL3365003 0.67 TAAR1 (0.50) NISCHALDH1A1KDM4EMAPTPOLB
SCHEMBL394300 0.66 TAAR1 (0.76) ALDH1A1KDM4EMAPTPOLBMEN1
SCHEMBL27397905 0.64 NISCH (0.53) NISCHALDH1A1KDM4EMAPTPOLB
SCHEMBL11974601 0.64 ALDH1A1 (0.52) ALDH1A1KDM4EMAPTPOLBMEN1
SCHEMBL11974593 0.64 ALDH1A1 (0.52) ALDH1A1KDM4EMAPTPOLBMEN1
SCHEMBL11974594 0.64 ALDH1A1 (0.52) ALDH1A1KDM4EMAPTPOLBMEN1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20050282740-A1 Methods and compositions for regulating protein-protein interactions LU KUN P 2005-12-22 US disclosed
EP-1028946-A1 INDAZOLE BIOISOSTERE REPLACEMENT OF CATECHOL IN THERAPEUTICALLY ACTIVE COMPOUNDS Pfizer Products Inc. (US) 2000-08-23 EP disclosed
WO-1999023077-A1 INDAZOLE BIOISOSTERE REPLACEMENT OF CATECHOL IN THERAPEUTICALLY ACTIVE COMPOUNDS PFIZER PRODUCTS INC. (US) 1999-05-14 WO disclosed