SCHEMBL6909709

SCHEMBL6909709

c1coc([C]2NCCO2)c1

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NISCH Q9Y2I1 1/20 0.46
ALDH1A1 P00352 5/20 0.39
MEN1 O00255 3/20 0.39
KMT2A Q03164 3/20 0.39
KDM4E B2RXH2 4/20 0.39
POLB P06746 3/20 0.39
HPGD P15428 3/20 0.39
MAPT P10636 2/20 0.39
PKM P14618 2/20 0.39
ALOX15 P16050 2/20 0.39
CASP1 P29466 2/20 0.39
PTPN7 P35236 2/20 0.39
RECQL P46063 2/20 0.39
BLM P54132 2/20 0.39
CASP7 P55210 2/20 0.39
HSD17B10 Q99714 2/20 0.39
TDP1 Q9NUW8 2/20 0.39
L3MBTL1 Q9Y468 2/20 0.39
USP2 O75604 1/20 0.39
LMNA P02545 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6519271 0.70 NISCH (0.52) NISCHALDH1A1MEN1KMT2AKDM4E
SCHEMBL1171231 0.68 NISCH (0.38) NISCHALDH1A1MEN1KMT2AKDM4E
SCHEMBL1799678 0.67 ALDH1A1 (0.63) NISCHALDH1A1MEN1KMT2AKDM4E
SCHEMBL6462643 0.65 ALDH1A1 (0.40) NISCHALDH1A1MEN1KMT2AKDM4E
SCHEMBL7229227 0.64 HPGDS (0.33) ADRA1AADRA1BADRA1D
SCHEMBL6911489 0.64 GRM5 (0.33) ADRA1AADRA1BADRA1D
SCHEMBL4398715 0.63 KDM4E (0.48) NISCHALDH1A1KDM4EPOLBHPGD
SCHEMBL6910633 0.63 NISCH (0.44) NISCHALDH1A1MEN1KMT2AKDM4E
SCHEMBL7367387 0.63 CHRM1 (0.33) ALDH1A1MAPTHSD17B10NPC1RAB9A
SCHEMBL1607474 0.63 NISCH (0.44) NISCHALDH1A1MEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 62 patents — showing the first 20. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0802732-B1 HERBICIDAL COMPOSITIONS OF 4-BENZOYLISOXAZOLE OR 2-CYANO-1,3-DIONE HERBICIDES AND ANTIDOTES THEREFOR ZENECA LTD (GB) 2000-04-19 EP claimed
WO-2000011954-A1 HERBICIDAL METHOD AVENTIS CROPSCIENCE S.A. (FR) 2000-03-09 WO claimed
EP-0565593-B1 REDUCING PESTICIDAL INTERACTIONS IN CROPS MONSANTO CO (US) 1999-03-03 EP claimed
EP-0802732-A1 HERBICIDAL COMPOSITIONS OF 4-BENZOYLISOXAZOLE OR 2-CYANO-1,3-DIONE HERBICIDES AND ANTIDOTES THEREFOR ZENECA LIMITED (GB) 1997-10-29 EP claimed
WO-1996021357-A1 HERBICIDAL COMPOSITIONS OF 4-BENZOYLISOXAZOLE OR 2-CYANO-1,3-DIONE HERBICIDES AND ANTIDOTES THEREFOR ZENECA LIMITED (GB) 1996-07-18 WO claimed
US-5536700-A Herbicidal compositions comprising aryl-5-haloalkylpyrazoles and glyphosate, it's salts, diquat or paraquat MONSANTO COMPANY (US) 1996-07-16 US claimed
EP-0603240-A1 SAFENING HERBICIDAL PYRAZOLYLSULFONYLURES MONSANTO COMPANY (US) 1994-06-29 EP claimed
US-5281571-A Herbicidal benzoxazinone- and benzothiazinone-substituted pyrazoles MONSANTO COMPANY (US) 1994-01-25 US claimed
US-5201933-A Haloacetamides MONSANTO COMPANY (US) 1993-04-13 US claimed
EP-0531271-A1 Safening herbicidal pyrazolysulfonylureas MONSANTO COMPANY (US) 1993-03-10 EP claimed
WO-1993003615-A1 SAFENING HERBICIDAL PYRAZOLYLSULFONYLURES MONSANTO COMPANY (US) 1993-03-04 WO claimed
WO-1992010098-A1 SAFENED HERBICIDAL SULFONAMIDE COMPOSITIONS MONSANTO COMPANY (US) 1992-06-25 WO claimed
EP-0480902-A1 Safening herbicidal benzoic acid derivatives MONSANTO COMPANY (US) 1992-04-15 EP claimed
EP-0436483-A2 Safening imidazolinone herbicides MONSANTO COMPANY (US) 1991-07-10 EP claimed
EP-0791571-B1 Benzoyl derivatives BAYER CROPSCIENCE AG (DE) 2004-06-16 EP disclosed
EP-1097117-A2 ARYL VINYL ETHER DERIVATIVES AND THEIR USE AS HERBICIDES AVENTIS AGRICULTURE LTD. (GB) 2001-05-09 EP disclosed
US-6121458-A ACYLATION, HALOGENATION, ALKYLATION, CATALYTIC OXIDATION, AND ESTERIFICATION; CYCLIZATION AND CONDENSATION WITH HYDRAZINE MONSANTO COMPANY (US) 2000-09-19 US disclosed
EP-0480902-A1 Safening herbicidal benzoic acid derivatives MONSANTO COMPANY (US) 1992-04-15 EP disclosed
WO-1992002509-A1 HERBICIDAL SUBSTITUTED ARYL ALKYLSULFONYL PYRAZOLES MONSANTO COMPANY (US) 1992-02-20 WO disclosed
EP-0436483-A2 Safening imidazolinone herbicides MONSANTO COMPANY (US) 1991-07-10 EP disclosed