SCHEMBL6520890

SCHEMBL6520890

Cc1[nH]c2cc(F)ccc2c1CCN

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR1D P28221 2/20 0.55
HTR6 P50406 2/20 0.55
CYP1A2 P05177 1/20 0.55
CYP3A4 P08684 1/20 0.55
CYP2D6 P10635 1/20 0.55
CYP2C9 P11712 1/20 0.55
MAPK1 P28482 1/20 0.55
CYP2C19 P33261 1/20 0.55
HTR7 P34969 1/20 0.55
HTR3A P46098 1/20 0.55
HSD17B10 Q99714 1/20 0.55
TDP1 Q9NUW8 1/20 0.55
PTGS1 P23219 2/20 0.50
PTGS2 P35354 2/20 0.50
HTR2A P28223 2/20 0.50
RAD52 P43351 1/20 0.46
BLM P54132 1/20 0.46
NPSR1 Q6W5P4 1/20 0.46
IDO1 P14902 1/20 0.45
TRPM8 Q7Z2W7 2/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL21546046 0.98 HTR1D (0.54) HTR1DHTR6CYP1A2CYP3A4CYP2D6
SCHEMBL8244089 0.87 HTR6 (0.68) HTR1DHTR6CYP1A2CYP3A4CYP2D6
Hydrochloric Acid SCHEMBL21546038 0.86 HTR6 (0.66) HTR1DHTR6CYP1A2CYP3A4CYP2D6
Cyanide SCHEMBL28561259 0.83 HTR6 (0.62) HTR1DHTR6CYP1A2CYP3A4CYP2D6
SCHEMBL21082250 0.81 PTGS1 (0.53) HSD17B10PTGS1PTGS2HTR2ASMN1; SMN2
SCHEMBL18235619 0.79 HTR6 (0.56) HTR1DHTR6CYP1A2CYP3A4CYP2D6
SCHEMBL29415611 0.76 ALDH1A1 (0.69) HTR1DHTR6CYP1A2CYP3A4CYP2D6
SCHEMBL1424220 0.76 ALDH1A1 (0.69) HTR1DHTR6CYP1A2CYP3A4CYP2D6
SCHEMBL31381374 0.75 KDM4E (0.63) CYP1A2CYP3A4CYP2C19PTGS1PTGS2
Hydrochloric Acid SCHEMBL273338 0.75 ALDH1A1 (0.67) HTR1DHTR6CYP1A2CYP3A4CYP2D6

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2018106907-A1 FUSED BICYCLIC ALKYLENE LINKED IMIDODICARBONIMIDIC DIAMIDES, METHODS FOR SYNTHESIS, AND USES IN THERARY NOVATARG, INC. (US) 2018-06-14 WO disclosed
EP-1532153-A1 AZEPINOINDOLE AND PYRIDOINDOLE DERIVATIVES AS PHARMACEUTICAL AGENTS X-Ceptor Therapeutics, Inc. (US) 2005-05-25 EP disclosed
WO-2003099821-A1 AZEPINOINDOLE AND PYRIDOINDOLE DERIVATIVES AS PHARMACEUTICAL AGENTS X-CEPTOR THERAPEUTICS, INC. (US) 2003-12-04 WO disclosed