Bromide

Bromide

SCHEMBL6522067

Br.Br.C=C1N(Cc2ccc(CN3C(=C)C(C)(C)c4ccccc43)cc2)c2ccccc2C1(C)C

nearest known ligand 0.59

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ACHEADRA1AADRA1BADRA1DADRA2AADRA2BADRA2CADRB1ADRB2ADRB3APH1AAPH1BCHRM2CHRM3EZH2GRIN2AHTR1AHTR1BHTR1DHTR1FHTR3ANCSTNP2RY12PSEN1PSEN2PSENENSIGMAR1SLC6A2SLC6A3SLC6A4

The experimentally established mechanism targets of Bromide. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
P2RX1 P51575 1/20 0.47
P2RX3 P56373 1/20 0.47
P2RX4 Q99571 1/20 0.47
P2RX7 Q99572 1/20 0.47
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
KMT2A Q03164 1/20 0.43
SCN9A Q15858 7/20 0.43
ELANE P08246 1/20 0.42
ALDH1A1 P00352 6/20 0.41
MAPT P10636 2/20 0.39
TP53 P04637 1/20 0.38
NPSR1 Q6W5P4 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1372846 0.98 P2RX1 (0.49) P2RX1P2RX3P2RX4P2RX7CYP1A2
Bromide SCHEMBL4444724 0.95 P2RX1 (0.44) P2RX1P2RX3P2RX4P2RX7CYP1A2
SCHEMBL6524494 0.94 P2RX1 (0.45) P2RX1P2RX3P2RX4P2RX7CYP1A2
SCHEMBL4434283 0.94 P2RX1 (0.45) P2RX1P2RX3P2RX4P2RX7CYP1A2
SCHEMBL10723893 0.93 P2RX1 (0.55) P2RX1P2RX3P2RX4P2RX7CYP1A2
SCHEMBL12147169 0.91 P2RX1 (0.47) P2RX1P2RX3P2RX4P2RX7CYP1A2
SCHEMBL12147197 0.91 P2RX1 (0.47) P2RX1P2RX3P2RX4P2RX7CYP1A2
SCHEMBL1372776 0.91 SCN9A (0.44) P2RX1P2RX3P2RX4P2RX7CYP1A2
SCHEMBL8552517 0.88 SCN9A (0.54) SCN9AMAPT
SCHEMBL3225659 0.87 CHRM5 (0.48) P2RX1P2RX3P2RX4P2RX7CYP1A2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-20110059545-A1 TIME-TEMPERATURE INDICATOR BASED ON OLIGOMERIC SPIROAROMATICS FRESHPOINT HOLDINGS SA (CH) 2011-03-10 US disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20110059545-A1 TIME-TEMPERATURE INDICATOR BASED ON OLIGOMERIC SPIROAROMATICS CCND3, CCNT1, SCO2 P2RX1 2411/4885P2RX3 1143/4885P2RX4 2042/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.