SCHEMBL6525277

SCHEMBL6525277

O=C1COc2ccc(CCCN3CCN(c4ccc5ccccc5n4)CC3)cc2N1.O=C1COc2ccc(CCN3CCN(c4ccc5ccccc5n4)CC3)cc2N1

nearest known ligand 0.62

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
HTR1A P08908 18/20 0.62
HTR1D P28221 15/20 0.62
HTR1B P28222 15/20 0.62
SLC6A4 P31645 14/20 0.62
DRD2 P14416 4/20 0.60
HTR2A P28223 3/20 0.60
KCNH2 Q12809 2/20 0.60
HTR2C P28335 1/20 0.60
HTR2B P41595 1/20 0.60
DRD4 P21917 2/20 0.55
SLC6A2 P23975 1/20 0.52
SLC6A3 Q01959 1/20 0.52
DRD3 P35462 1/20 0.52

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4172034 0.98 HTR1A (0.64) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL4189338 0.96 HTR1A (0.66) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL4174687 0.85 HTR1A (0.61) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL4172085 0.82 HTR1A (0.53) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL532984 0.79 HTR1A (0.63) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL14510673 0.78 HTR1A (0.62) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL10864650 0.78 DRD2 (0.74) HTR1AHTR1DHTR1BSLC6A4DRD2
Hydrochloric Acid SCHEMBL2358961 0.77 HTR1A (0.73) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL4189187 0.77 HTR1A (1.00) HTR1AHTR1DHTR1BSLC6A4DRD2
SCHEMBL4182140 0.77 HTR1A (0.72) HTR1AHTR1DHTR1BSLC6A4DRD2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1562917-A1 BENZOXAZINONE DERIVATIVES, PREPARATION THEREOF AND USES IN THE TREATMENT OF CNS AND OTHER DISORDERS GLAXO GROUP LIMITED (GB) 2005-08-17 EP claimed
WO-2004046124-A1 BENZOXAZINONE DERIVATIVES, PREPARATION THEREOF AND USES IN THE TREATMENT OF CNS AND OTHER DISORDERS GLAXO GROUP LIMITED (GB) 2004-06-03 WO claimed