SCHEMBL6527339

SCHEMBL6527339

COc1ccc(N(c2ccc(-c3nn[nH]n3)cc2)C(O)c2cccnc2)cc1OC1CCCC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
PDE4A P27815 14/20 0.47
ALDH1A1 P00352 1/20 0.42
S1PR1 P21453 1/20 0.41
S1PR3 Q99500 1/20 0.41
PDE4D Q08499 8/20 0.40
PDE4B Q07343 7/20 0.40
PDE4C Q08493 7/20 0.40
XDH P47989 1/20 0.39
ADRB1 P08588 1/20 0.39
ADRB3 P13945 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6533002 0.94 PDE4A (0.46) PDE4AALDH1A1PDE4DPDE4BPDE4C
SCHEMBL6530112 0.90 PDE4A (0.42) PDE4AALDH1A1PDE4DPDE4BPDE4C
SCHEMBL6528128 0.86 ALDH1A1 (0.41) PDE4AALDH1A1PDE4DPDE4BPDE4C
SCHEMBL2924797 0.83 PDE4A (0.47) PDE4AALDH1A1S1PR1S1PR3PDE4D
SCHEMBL1157355 0.82 PDE4A (0.51) PDE4AALDH1A1S1PR1S1PR3PDE4D
SCHEMBL6465669 0.80 PDE4A (0.51) PDE4APDE4DPDE4BPDE4C
SCHEMBL6469266 0.79 PDE4A (0.49) PDE4APDE4DPDE4BPDE4C
SCHEMBL2924989 0.79 PDE4A (0.46) PDE4AALDH1A1PDE4DPDE4BPDE4C
SCHEMBL1157468 0.78 PDE4A (0.51) PDE4AALDH1A1PDE4DPDE4BPDE4C
SCHEMBL6469942 0.78 PDE4D (0.48) PDE4APDE4DPDE4BPDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1569908-A2 PYRIDINE N-OXIDE COMPOUNDS AS PHOSPHODIESTERASE 4 INHIBITORS Memory Pharmaceutical Corporation (US) 2005-09-07 EP disclosed
WO-2004046113-A2 PYRIDINE N-OXIDE COMPOUNDS AS PHOSPHODIESTERASE 4 INHIBITORS MEMORY PHARMACEUTICALS CORPORATION (US) 2004-06-03 WO disclosed