SCHEMBL6527610

SCHEMBL6527610

Cc1c(N2CCC(C)(CN(C)CCC#N)C2)c(F)cc2c(=O)c(C(=O)O)cn(C3CC3)c12

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KCNH2 Q12809 6/20 0.59
ALDH1A1 P00352 4/20 0.45
KDM4E B2RXH2 4/20 0.45
HPGD P15428 3/20 0.45
POLB P06746 2/20 0.45
OPRM1 P35372 2/20 0.45
HSD17B10 Q99714 2/20 0.45
PRKD3 O94806 1/20 0.45
ALOX15 P16050 1/20 0.45
CLK2 P49760 1/20 0.45
CLK4 Q9HAZ1 1/20 0.45
TDP1 Q9NUW8 1/20 0.45
CHRM2 P08172 1/20 0.44
CHRM1 P11229 1/20 0.44
OPRD1 P41143 1/20 0.44
TOP2A P11388 5/20 0.44
TOP2B Q02880 5/20 0.44
LMNA P02545 1/20 0.42
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528949 0.92 KCNH2 (0.57) KCNH2ALDH1A1KDM4EHPGDPOLB
SCHEMBL6529675 0.85 KCNH2 (0.44) KCNH2ALDH1A1KDM4EHPGDPOLB
SCHEMBL9377634 0.84 KCNH2 (0.55) KCNH2ALDH1A1KDM4EHPGDPOLB
SCHEMBL6527346 0.82 KCNH2 (0.68) KCNH2ALDH1A1KDM4EHPGDPOLB
SCHEMBL6528606 0.81 KCNH2 (0.60) KCNH2ALDH1A1KDM4EHPGDPOLB
SCHEMBL6529048 0.81 KCNH2 (0.66) KCNH2ALDH1A1KDM4EHPGDPOLB
SCHEMBL6529826 0.81 KCNH2 (0.64) KCNH2ALDH1A1KDM4EHPGDPOLB
SCHEMBL9377051 0.81 KCNH2 (0.56) KCNH2ALDH1A1KDM4EHPGDPOLB
SCHEMBL6528390 0.80 KCNH2 (0.56) KCNH2ALDH1A1KDM4EHPGDPOLB
SCHEMBL9377877 0.80 ALDH1A1 (0.62) KCNH2ALDH1A1KDM4EHPGDPOLB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005049602-A1 QUINOLONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2005-06-02 WO claimed
WO-2005051380-A1 SUBSTITUTED UREA-OCTAHYDROINDOLS AS ANTAGONISTS OF MELANIN CONCENTRATING HORMONE RECEPTOR 1 (MCH1R) BIOVITRUM AB (SE) 2005-06-09 WO disclosed
WO-2005049602-A1 QUINOLONE ANTIBACTERIAL AGENTS WARNER-LAMBERT COMPANY LLC (US) 2005-06-02 WO disclosed