Terazosin

Terazosin

SCHEMBL6528

COc1cc2nc(N3CCN(C(=O)C4CCCO4)CC3)nc(N)c2cc1OC

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Full drug profile on Sugi Atlas →

Known targets — ChEMBL curated mechanism

ADRA1AADRA1BADRA1D

The experimentally established mechanism targets of Terazosin. The predicted profile below is derived independently by chemical similarity — agreement is a validation signal, a miss is honest.

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ADRA1D known ✓ P25100 3/20 1.00
ADRA1A known ✓ P35348 3/20 1.00
ADRA1B known ✓ P35368 3/20 1.00
KDM4E B2RXH2 5/20 1.00
ALDH1A1 P00352 4/20 1.00
HPGD P15428 4/20 1.00
GLA P06280 4/20 1.00
HSD17B10 Q99714 3/20 1.00
GAA P10253 3/20 1.00
MAPK1 P28482 2/20 1.00
ADRA2A P08913 2/20 1.00
ADRA2B P18089 2/20 1.00
ADRA2C P18825 2/20 1.00
DRD1 P21728 2/20 1.00
OPRM1 P35372 2/20 1.00
OPRK1 P41145 2/20 1.00
KCNH2 Q12809 2/20 1.00
TP53 P04637 1/20 1.00
TSHR P16473 1/20 1.00
SLC22A1 O15245 1/20 1.00

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Terazosin SCHEMBL41546 1.00 KDM4E (1.00) KDM4EALDH1A1HPGDGLAHSD17B10
Terazosin SCHEMBL30684952 1.00 KDM4E (1.00) KDM4EALDH1A1HPGDGLAHSD17B10
Terazosin SCHEMBL5424458 1.00 KDM4E (1.00) KDM4EALDH1A1HPGDGLAHSD17B10
Terazosin SCHEMBL41545 0.99 KDM4E (1.00) KDM4EALDH1A1HPGDGLAHSD17B10
Terazosin SCHEMBL5427410 0.99 KDM4E (1.00) KDM4EALDH1A1HPGDGLAHSD17B10
Terazosin SCHEMBL31284920 0.99 KDM4E (1.00) KDM4EALDH1A1HPGDGLAHSD17B10
Terazosin SCHEMBL8057933 0.99 KDM4E (0.98) KDM4EALDH1A1HPGDGLAHSD17B10
Terazosin SCHEMBL5525882 0.99 KDM4E (1.00) KDM4EALDH1A1HPGDGLAHSD17B10
Terazosin SCHEMBL9053035 0.98 KDM4E (1.00) KDM4EALDH1A1HPGDGLAHSD17B10
Terazosin SCHEMBL1133792 0.98 KDM4E (0.96) KDM4EALDH1A1HPGDGLAHSD17B10

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Appears in 20351 patents — a generic fragment claimed broadly, so it's down-weighted as IP noise. Top by claim status then date:

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4727545-A2 COMBINATION TREATMENTS FOR DEPRESSION AND OTHER DISORDERS Neurawell Therapeutics (US) 2026-04-22 EP claimed
EP-4724049-A1 MODIFIED RELEASE FILL COMPOSITIONS FOR DOSAGE FORMS AND METHODS OF PREPARATION AND USE THEREOF Catalent Ontario Limited (CA) 2026-04-15 EP claimed
US-12599554-B2 Pharmaceutical formulations comprising tadalafil KYDES PHARMACEUTICALS LLC (US) 2026-04-14 US claimed
US-12569575-B2 Radiopaque particle compositions and uses thereof GUSTAVE ROUSSY TRANSFERT (FR) 2026-03-10 US claimed
US-20250375376-A1 STABLE ORAL LIQUID COMPOSITION OF TERAZOSIN Novitium Pharma LLC (US) 2025-12-11 US claimed
US-20250367321-A1 COMPOSITIONS AND METHODS INVOLVING ADGRG6 THE REGENTS OF THE UNIVERSITY OF CALIFORNIA (US) 2025-12-04 US claimed
EP-3699174-B1 COMPOSITION FOR PREVENTING OR TREATING TNF-RELATED DISEASES, CONTAINING DERIVATIVE AS ACTIVE INGREDIENT, AND METHOD FOR INHIBITING TNF ACTIVITY BY USING SAME ILAB (KR) 2025-11-12 EP claimed
US-20250319068-A1 TREATMENT OF DISEASES VIA ADMINISTRATION OF BUNTANETAP AND AN ANTIHYPERTENSIVE AGENT ANNOVIS BIO, INC. (US) 2025-10-16 US claimed
US-20250302887-A1 AMMONIA OXIDIZING MICROORGANISMS FOR THE REGULATION OF BLOOD PRESSURE AOBIOME LLC (US) 2025-10-02 US claimed
US-12427108-B2 Stable oral liquid composition of terazosin Novitium Pharma LLC (US) 2025-09-30 US claimed
EP-0526001-A1 Substituted triazolinones MERCK & CO. INC. (US) 1993-02-03 EP claimed
WO-1993001177-A1 SUBSTITUTED TRIAZOLINONES MERCK & CO., INC. (US) 1993-01-21 WO claimed
WO-1992016213-A1 PHARMACEUTICAL COMBINATION FOR THE TREATMENT OF PROSTATIC HYPERPLASIA, CONTAINING A 5 ALPHA-REDUCTASE INHIBITOR AND AN ANTIANDROGEN MERCK & CO., INC. (US) 1992-10-01 WO claimed
WO-1992014453-A1 COMPOSITIONS AND METHODS OF TREATMENT OF SYMPATHETICALLY MAINTAINED PAIN ARC 1, INC. (US) 1992-09-03 WO claimed
WO-1992011851-A1 METHOD AND COMPOSITIONS FOR TREATMENT OF SEXUAL IMPOTENCE LARAGH JOHN H (US) 1992-07-23 WO claimed
WO-1992000073-A1 R(+)-TERAZOSIN ABBOTT LABORATORIES (US) 1992-01-09 WO claimed
EP-0430287-A2 Sustained-release drug dosage units ABBOTT LABORATORIES (US) 1991-06-05 EP claimed
EP-0189336-A1 Pharmaceutical compositions containing an alpha-blocker and a calcium antagonist SYNTHELABO (FR) 1986-07-30 EP claimed
US-4112097-A QUINAZOLINES ABBOTT LABORATORIES (US) 1978-09-05 US claimed
US-4026894-A 2(4(TETRAHYDRO-2-FUROYL)-PIPERAZINO)-4-AMINO-6,7-DIMETHOXYQUINAZOLINE OR 2-(4(TETRAHYDROPYRAN-2-CARBONYL)-PIPERAZINYL)-4-AMINO-6,7 -DIMETHOXYQUINAZOLINE ABBOTT LABORATORIES (US) 1977-05-31 US claimed