SCHEMBL6528748

SCHEMBL6528748

COc1ccc(CN(C)C)cc1-c1cc(Nc2ccc3[nH]ncc3c2)ncn1

nearest known ligand 0.48

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
RET P07949 1/20 0.48
CCNT1 O60563 10/20 0.46
CDK9 P50750 10/20 0.46
ROCK2 O75116 2/20 0.46
AGPAT2 O15120 1/20 0.46
IGF1R P08069 1/20 0.46
KDR P35968 2/20 0.43
USP2 O75604 1/20 0.43
ALDH1A1 P00352 1/20 0.43
LMNA P02545 1/20 0.43
CYP1A2 P05177 1/20 0.43
CYP2D6 P10635 1/20 0.43
ALOX15 P16050 1/20 0.43
CYP2C19 P33261 1/20 0.43
HSD17B10 Q99714 1/20 0.43
CLK4 Q9HAZ1 1/20 0.43
ROCK1 Q13464 1/20 0.43
EGFR P00533 1/20 0.42
TNIK Q9UKE5 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6531053 0.84 ROCK2 (0.46) RETROCK2KDRUSP2ALDH1A1
SCHEMBL4104723 0.83 USP2 (0.64) RETCCNT1CDK9USP2ALDH1A1
SCHEMBL6531231 0.81 ROCK2 (0.47) CCNT1CDK9ROCK2ROCK1EGFR
SCHEMBL4116187 0.75 USP2 (0.64) RETCCNT1CDK9AGPAT2IGF1R
SCHEMBL6530116 0.74 TNIK (0.46) ROCK2KDRUSP2ALDH1A1LMNA
SCHEMBL15486390 0.72 CYP1A2 (0.66) CCNT1CDK9USP2ALDH1A1LMNA
SCHEMBL6530951 0.72 MKNK1 (0.51) ROCK2KDREGFRTNIK
SCHEMBL6531731 0.72 TNIK (0.49) ROCK2KDREGFRTNIK
SCHEMBL30611394 0.72 ROCK2 (0.58) RETROCK2KDRROCK1EGFR
SCHEMBL6530590 0.72 ABL1 (0.60) RETROCK2KDRROCK1EGFR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005103036-A1 PYRIMIDIN-4-YL-1H-INDAZOL-5YL-AMINES AS CHK1 KINASES INHIBITORS BIOFOCUS DISCOVERY LTD (GB) 2005-11-03 WO claimed
WO-2005082892-A2 TRIAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S LABORATORIES LTD. (IN) 2005-09-09 WO disclosed