SCHEMBL6528847

SCHEMBL6528847

COc1ccc(Sc2nc(Nc3cccc(F)c3)nc(N[C@@H](CC(C)C)C(N)=O)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
SYK P43405 8/20 0.43
KCNH3 Q9ULD8 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
SCN9A Q15858 2/20 0.40
FPR2 P25090 1/20 0.40
ALDH1A1 P00352 1/20 0.39
CYP1A2 P05177 1/20 0.39
CYP2D6 P10635 1/20 0.39
CYP2C9 P11712 1/20 0.39
CYP2C19 P33261 1/20 0.39
L3MBTL1 Q9Y468 1/20 0.39
CTSK P43235 1/20 0.39
CHRNA7 P36544 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528931 0.93 KCNH3 (0.41) KCNH3MEN1KMT2AALDH1A1CYP1A2
SCHEMBL6508192 0.93 KCNH3 (0.41) KCNH3MEN1KMT2AALDH1A1CYP1A2
SCHEMBL6508189 0.93 KCNH3 (0.41) KCNH3MEN1KMT2AALDH1A1CYP1A2
SCHEMBL6532662 0.87 CTSK (0.42) KCNH3ALDH1A1CYP1A2CYP2D6CYP2C9
SCHEMBL6531457 0.87 ATM (0.45) KCNH3ALDH1A1CTSK
SCHEMBL6530634 0.87 CTSK (0.45) KCNH3ALDH1A1CTSK
SCHEMBL6530404 0.86 IDH2 (0.43) KCNH3MEN1KMT2AALDH1A1CYP1A2
SCHEMBL6527570 0.86 IDH2 (0.43) KCNH3MEN1KMT2AALDH1A1CYP1A2
SCHEMBL6530873 0.85 MAPT (0.41) MEN1KMT2AALDH1A1CTSK
SCHEMBL6528746 0.85 CTSK (0.44) KCNH3MEN1KMT2ACTSK

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed