SCHEMBL6529174

SCHEMBL6529174

COc1ccccc1Cn1cnc(C)c1

nearest known ligand 0.47

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.47
KDM4E B2RXH2 2/20 0.47
TDP1 Q9NUW8 1/20 0.47
DBH P09172 1/20 0.44
LMNA P02545 3/20 0.44
HTT P42858 2/20 0.44
NPSR1 Q6W5P4 1/20 0.44
QPCT Q16769 1/20 0.43
GAA P10253 1/20 0.42
MAPT P10636 1/20 0.42
P2RX7 Q99572 1/20 0.42
GNAI3 P08754 1/20 0.42
USP2 O75604 1/20 0.42
CYP2D6 P10635 1/20 0.42
PHF8 Q9UPP1 1/20 0.42
TSHR P16473 1/20 0.42
L3MBTL1 Q9Y468 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6530474 0.83 ALDH1A1 (0.43) ALDH1A1KDM4ETDP1DBHLMNA
SCHEMBL6529662 0.78 PHF8 (0.54) ALDH1A1LMNAHTTGAAPHF8
SCHEMBL8336583 0.73 CYP19A1 (0.68) ALDH1A1QPCTMAPTCYP2D6
SCHEMBL3726218 0.73 CYP19A1 (0.54) ALDH1A1KDM4ETDP1MAPT
SCHEMBL16549376 0.73 QPCT (0.38) ALDH1A1KDM4ELMNAQPCTGAA
SCHEMBL6530144 0.71 CDK5 (0.51) ALDH1A1KDM4EQPCTGAAMAPT
SCHEMBL3976264 0.70 GAA (0.47) ALDH1A1DBHLMNAGAAMAPT
SCHEMBL19157912 0.70 PHF8 (0.42) QPCTP2RX7PHF8
SCHEMBL8066986 0.69 PSEN1 (0.51)
SCHEMBL15929449 0.69 ALDH1A1 (0.51) ALDH1A1KDM4ETDP1DBHLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO claimed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed