SCHEMBL6530058

SCHEMBL6530058

COC(=O)c1ccc(NC(=O)Nc2ccc(-c3nc4ccccc4[nH]3)cc2)cc1

nearest known ligand 0.83

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.83
RAB9A P51151 2/20 0.83
KDM4E B2RXH2 2/20 0.83
ALDH1A1 P00352 2/20 0.83
LMNA P02545 1/20 0.83
PKM P14618 1/20 0.83
HPGD P15428 1/20 0.83
NFKB1 P19838 1/20 0.83
NFKB2 Q00653 1/20 0.83
RELA Q04206 1/20 0.83
SMN1; SMN2 Q16637 1/20 0.83
HPSE Q9Y251 10/20 0.79
MMP2 P08253 3/20 0.65
MMP9 P14780 3/20 0.65
MMP8 P22894 3/20 0.65
MMP13 P45452 3/20 0.65
MEN1 O00255 1/20 0.61
KMT2A Q03164 1/20 0.61
TNKS O95271 1/20 0.60

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2617471 0.91 NPC1 (1.00) NPC1RAB9AKDM4EALDH1A1LMNA
SCHEMBL6533676 0.89 HPSE (1.00) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL943034 0.89 HPSE (1.00) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL6530157 0.85 HPSE (0.77) NPC1RAB9AKDM4EALDH1A1LMNA
SCHEMBL6532513 0.85 HPSE (0.87) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL6528576 0.84 HPSE (0.82) NPC1RAB9AKDM4EALDH1A1PKM
SCHEMBL16147815 0.83 KMT2A (0.69) NPC1RAB9AKDM4EALDH1A1LMNA
SCHEMBL6506260 0.83 MMP2 (0.93) NPC1RAB9AKDM4EALDH1A1HPGD
SCHEMBL25674602 0.83 HPSE (0.78) NPC1RAB9AKDM4EALDH1A1LMNA
SCHEMBL6529336 0.83 HPSE (0.73) NPC1RAB9AKDM4EALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005042495-A1 (BENZIMIDAZOL-2-YL)-PHENYL-PHENYL-UREA COMPOUNDS AND METHODS FOR INHIBITING HEPARANASE ACTIVITY IMCLONE SYSTEMS INCORPORATED (US) 2005-05-12 WO disclosed