SCHEMBL6530135

SCHEMBL6530135

[CH2]c1cn(Cc2ccc(OC)cc2)cn1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CDK5 Q00535 1/20 0.50
CDK5R1 Q15078 1/20 0.50
CYP19A1 P11511 2/20 0.48
ALDH1A1 P00352 2/20 0.45
KDM4E B2RXH2 1/20 0.45
MAPT P10636 1/20 0.45
ALOX15 P16050 1/20 0.45
CMA1 P23946 1/20 0.45
HSP90AA1 P07900 1/20 0.43
KDM4C Q9H3R0 1/20 0.43
KDM5B Q9UGL1 1/20 0.43
CYP11B1 P15538 1/20 0.43
GSK3A P49840 1/20 0.42
GSK3B P49841 1/20 0.42
SIGMAR1 Q99720 1/20 0.41
SMN1; SMN2 Q16637 2/20 0.41
LMNA P02545 1/20 0.41
MEN1 O00255 1/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6530144 0.82 CDK5 (0.51) CDK5CDK5R1CYP19A1ALDH1A1KDM4E
SCHEMBL27744436 0.82 CDK5 (0.51) CDK5CDK5R1CYP19A1ALDH1A1KDM4E
SCHEMBL6528479 0.82 LPO (0.51) CYP19A1ALDH1A1KDM4EMAPTCMA1
SCHEMBL7510401 0.81 CDK5 (0.50) CDK5CDK5R1CYP19A1ALDH1A1KDM4E
SCHEMBL2979842 0.81 CDK5 (0.50) CDK5CDK5R1CYP19A1ALDH1A1KDM4E
SCHEMBL15707234 0.81 CDK5 (0.50) CDK5CDK5R1CYP19A1ALDH1A1KDM4E
SCHEMBL6531582 0.80 CYP11B1 (0.49) CYP19A1ALDH1A1KDM4EKDM4CKDM5B
SCHEMBL5761329 0.79 CYP11B1 (0.54) CDK5CDK5R1ALDH1A1MAPTHSP90AA1
SCHEMBL1196868 0.78 HPGDS (0.51) CDK5CDK5R1CYP19A1MAPTKDM4C
SCHEMBL17982242 0.77 CDK5 (0.53) CDK5CDK5R1CYP19A1ALDH1A1KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO claimed
WO-2005016883-A2 ACRYLAMIDE DERIVATIVES AS VLA-1 INTEGRIN ANTAGONISTS AND USES THEREOF ICOS CORPORATION (US) 2005-02-24 WO disclosed