SCHEMBL6530216

SCHEMBL6530216

COc1ccc(Sc2nc(Nc3cccc(F)c3)nc(N(CCCN3CCCC3=O)C(=O)[C@@H](N)CC(C)C)n2)cc1

nearest known ligand 0.38

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 2/20 0.38
RAB9A P51151 1/20 0.38
EGFR P00533 8/20 0.38
ITK Q08881 5/20 0.37
SMN1; SMN2 Q16637 1/20 0.37
ATM Q13315 1/20 0.37
HSD17B10 Q99714 4/20 0.36
ALDH1A1 P00352 3/20 0.36
HPGD P15428 3/20 0.36
MAPK1 P28482 3/20 0.36
KDM4E B2RXH2 2/20 0.36
USP2 O75604 2/20 0.36
NPSR1 Q6W5P4 1/20 0.36
RCE1 Q9Y256 1/20 0.35
GALR2 O43603 1/20 0.35
GAA P10253 1/20 0.35
TSHR P16473 1/20 0.35
CASP1 P29466 1/20 0.35
CASP7 P55210 1/20 0.35
POLB P06746 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528784 0.88 GALR2 (0.37) GALR2POLB
SCHEMBL6528279 0.88 GALR2 (0.38) GALR2
SCHEMBL6528181 0.87 TBK1 (0.35) ALDH1A1HPGDMAPK1POLB
SCHEMBL6529648 0.86 PDPK1 (0.41) EGFRMAPK1USP2TSHRPOLB
SCHEMBL6528749 0.83 MEN1 (0.37) ALDH1A1HPGDMAPK1POLB
SCHEMBL6531461 0.81 EGFR (0.39) EGFRALDH1A1HPGDPOLB
SCHEMBL6530210 0.81 NPC1 (0.45) NPC1RAB9AEGFRITKSMN1; SMN2
SCHEMBL6533478 0.81 ITK (0.36) NPC1RAB9AEGFRITKSMN1; SMN2
SCHEMBL6529551 0.80 CHRNA7 (0.35) ALDH1A1MAPK1KDM4EPOLB
SCHEMBL6530876 0.80 MAPT (0.38) RAB9AEGFRSMN1; SMN2ALDH1A1HPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed