SCHEMBL6528181

SCHEMBL6528181

COCCCN(C(=O)[C@@H](N)CC(C)C)c1nc(Nc2cccc(F)c2)nc(Sc2ccc(OC)cc2)n1

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
TBK1 Q9UHD2 1/20 0.35
CFTR P13569 2/20 0.35
TP53 P04637 1/20 0.34
POLB P06746 1/20 0.34
MAPT P10636 1/20 0.34
MEN1 O00255 3/20 0.34
KMT2A Q03164 3/20 0.34
RAD52 P43351 1/20 0.34
SCN9A Q15858 1/20 0.34
BTK Q06187 1/20 0.33
CHRNA7 P36544 1/20 0.33
MAPK1 P28482 1/20 0.33
HTT P42858 1/20 0.33
AURKB Q96GD4 1/20 0.33
CDC7 O00311 1/20 0.33
CDK19 Q9BWU1 1/20 0.33
SYK P43405 2/20 0.32
HPGD P15428 1/20 0.32
ALDH1A1 P00352 1/20 0.32
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6528749 0.90 MEN1 (0.37) CFTRTP53POLBMAPTMEN1
SCHEMBL6528784 0.87 GALR2 (0.37) CFTRPOLBSYKCYP1A2CYP2D6
SCHEMBL6531461 0.87 EGFR (0.39) CFTRTP53POLBMAPTMEN1
SCHEMBL6528279 0.87 GALR2 (0.38) SYKCYP1A2CYP2D6CYP2C19
SCHEMBL6530216 0.87 NPC1 (0.38) POLBMAPK1HPGDALDH1A1
SCHEMBL6533478 0.86 ITK (0.36) CFTRTP53POLBMAPTMEN1
SCHEMBL6529648 0.86 PDPK1 (0.41) POLBMEN1KMT2ABTKMAPK1
SCHEMBL6528183 0.86 TBK1 (0.34) TBK1CFTRTP53POLBMAPT
SCHEMBL6529551 0.86 CHRNA7 (0.35) CFTRTP53POLBMAPTMEN1
SCHEMBL6530876 0.85 MAPT (0.38) POLBMAPTMEN1KMT2AMAPK1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005003103-A2 2, 4, 6-TRI-SUBSTITUTED 6-MEMBERED HETEROCYCLES AND THEIR USE IN THE TREATMENT OF NEURODEGENERATIVE DISEASES ASTRAZENECA AB (SE) 2005-01-13 WO disclosed