SCHEMBL6530375

SCHEMBL6530375

CN(C)c1cc(-c2cccc(F)c2)nc2ccc(Br)cc12.CN(C)c1cc(-c2cccc(F)c2)nc2ccccc12

nearest known ligand 0.49

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
ACP1 P24666 3/20 0.49
ABCG2 Q9UNQ0 2/20 0.44
RXFP1 Q9HBX9 2/20 0.42
ADORA2A P29274 2/20 0.41
KDM4E B2RXH2 1/20 0.39
HPGD P15428 1/20 0.39
NPSR1 Q6W5P4 1/20 0.39
POLB P06746 1/20 0.39
PRNP P04156 1/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
PTGFR P43088 2/20 0.38
MEN1 O00255 1/20 0.38
MAPT P10636 1/20 0.38
KMT2A Q03164 1/20 0.38
CYP19A1 P11511 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4025078 0.95 RXFP1 (0.42) ACP1ABCG2RXFP1ADORA2AKDM4E
SCHEMBL4825593 0.90 ACP1 (0.57) ACP1ABCG2ADORA2AHPGDALDH1A1
SCHEMBL4823939 0.81 KMT2A (0.49) ACP1RXFP1ADORA2AKDM4EPRNP
SCHEMBL4031738 0.81 DHODH (0.45) ACP1ABCG2ADORA2AMEN1KMT2A
SCHEMBL4823424 0.81 MAP4K4 (0.43) ACP1ABCG2ADORA2AKDM4EHPGD
SCHEMBL4026356 0.79 NT5E (0.43) ACP1ABCG2ADORA2AKDM4EHPGD
SCHEMBL4032316 0.78 CYP1A2 (0.46) ACP1ABCG2RXFP1ADORA2AKDM4E
SCHEMBL6001448 0.78 ACP1 (0.68) ACP1ADORA2AKDM4EHPGDALDH1A1
SCHEMBL4025761 0.77 NT5E (0.44) ACP1ABCG2RXFP1ADORA2AKDM4E
SCHEMBL4028750 0.77 ABCG2 (0.48) ACP1ABCG2RXFP1KDM4EHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6906193-B2 N-type calcium channel antagonists for the treatment of pain ASTRAZENECA AB (SE) 2005-06-14 US disclosed