SCHEMBL4031738

SCHEMBL4031738

CN(C)c1cc(-c2cccc(F)c2)nc2ccc(-c3ccc(F)cc3)cc12

nearest known ligand 0.45

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 3/20 0.45
NT5E P21589 2/20 0.45
ACP1 P24666 2/20 0.44
MAP4K4 O95819 2/20 0.42
ADORA2A P29274 1/20 0.41
MEN1 O00255 1/20 0.40
KMT2A Q03164 1/20 0.40
TOP1 P11387 1/20 0.40
ABCG2 Q9UNQ0 2/20 0.39
TAAR1 Q96RJ0 1/20 0.39
ESR2 Q92731 1/20 0.39
ROCK2 O75116 1/20 0.38
CDC7 O00311 1/20 0.38
PIM1 P11309 1/20 0.38
GSK3B P49841 1/20 0.38
HIPK2 Q9H2X6 1/20 0.38
CLK4 Q9HAZ1 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4026356 0.93 NT5E (0.43) DHODHNT5EACP1MAP4K4ADORA2A
SCHEMBL4027654 0.89 ACP1 (0.48) DHODHNT5EACP1MEN1KMT2A
SCHEMBL4025761 0.88 NT5E (0.44) DHODHNT5EACP1MAP4K4ADORA2A
SCHEMBL4022559 0.87 NT5E (0.49) DHODHNT5EACP1MAP4K4ABCG2
SCHEMBL4025213 0.86 DHFR (0.44) DHODHNT5EACP1MAP4K4MEN1
SCHEMBL4823424 0.85 MAP4K4 (0.43) DHODHNT5EACP1MAP4K4ADORA2A
SCHEMBL4025078 0.85 RXFP1 (0.42) ACP1MAP4K4ADORA2AKMT2AABCG2
SCHEMBL4032316 0.84 CYP1A2 (0.46) DHODHNT5EACP1ADORA2AABCG2
SCHEMBL4031533 0.84 LMNA (0.47) DHODHADORA2AMEN1KMT2ACLK4
SCHEMBL4026216 0.84 FYN (0.46) NT5EACP1MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339690-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2009-01-21 EP disclosed