SCHEMBL4026356

SCHEMBL4026356

Cc1ccc(-c2ccc3nc(-c4cccc(F)c4)cc(N(C)C)c3c2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NT5E P21589 2/20 0.43
ACP1 P24666 2/20 0.43
ADORA2A P29274 1/20 0.42
DHODH Q02127 4/20 0.42
MAP4K4 O95819 1/20 0.40
MAPT P10636 2/20 0.40
HPGD P15428 2/20 0.40
MEN1 O00255 2/20 0.40
KMT2A Q03164 2/20 0.40
KDM4E B2RXH2 1/20 0.40
ALDH1A1 P00352 1/20 0.40
TDP1 Q9NUW8 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
MGAM O43451 1/20 0.39
GAA P10253 1/20 0.39
SI P14410 1/20 0.39
MGAM2 Q2M2H8 1/20 0.39
HSP90AA1 P07900 1/20 0.38
ALOX15 P16050 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4031738 0.93 DHODH (0.45) NT5EACP1ADORA2ADHODHMAP4K4
SCHEMBL4027654 0.87 ACP1 (0.48) NT5EACP1DHODHMAPTHPGD
SCHEMBL4032316 0.85 CYP1A2 (0.46) NT5EACP1ADORA2ADHODHHPGD
SCHEMBL4022559 0.85 NT5E (0.49) NT5EACP1DHODHMAP4K4TDP1
SCHEMBL4025213 0.84 DHFR (0.44) NT5EACP1DHODHMAP4K4MEN1
SCHEMBL4025761 0.83 NT5E (0.44) NT5EACP1ADORA2ADHODHMAP4K4
SCHEMBL4025078 0.82 RXFP1 (0.42) ACP1ADORA2AMAP4K4HPGDKMT2A
SCHEMBL4823424 0.82 MAP4K4 (0.43) NT5EACP1ADORA2ADHODHMAP4K4
SCHEMBL4031533 0.82 LMNA (0.47) ADORA2ADHODHMAPTHPGDMEN1
SCHEMBL4026216 0.82 FYN (0.46) NT5EACP1HPGDMEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1339690-B1 N-TYPE CALCIUM CHANNEL ANTAGONISTS FOR THE TREATMENT OF PAIN ASTRAZENECA AB (SE) 2009-01-21 EP disclosed