SCHEMBL6530409

SCHEMBL6530409

CC(=S)NCc1cn(-c2cc(F)c(C3=CCN(C(=O)OC(C)(C)C)CC3)c(F)c2)nn1

nearest known ligand 0.54

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
GRM1 Q13255 11/20 0.54
GRM5 P41594 10/20 0.54
GPR119 Q8TDV5 3/20 0.46
KIT P10721 1/20 0.41
CA1 P00915 3/20 0.40
CA2 P00918 3/20 0.40
CA9 Q16790 3/20 0.40
CA12 O43570 2/20 0.40
CDK9 P50750 1/20 0.39
PDK4 Q16654 1/20 0.39
CA4 P22748 1/20 0.38
CA7 P43166 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6531659 0.93 GRM1 (0.54) GRM1GRM5GPR119KITCA1
SCHEMBL6530325 0.86 GRM1 (0.58) GRM1GRM5GPR119CDK9PDK4
SCHEMBL6529525 0.80 GRM1 (0.55) GRM1GRM5GPR119CDK9PDK4
SCHEMBL6529331 0.79 GRM1 (0.38) GRM1GRM5GPR119CA1CA2
SCHEMBL6530570 0.76 GRM1 (0.34) GRM1GRM5GPR119CDK9
SCHEMBL6918444 0.76 NOTUM (0.38)
SCHEMBL6922295 0.75 NOTUM (0.37)
SCHEMBL6510881 0.75 CA1 (0.43) GRM1GRM5GPR119CA1CA2
SCHEMBL6532521 0.74 NOTUM (0.46) GRM1GRM5
SCHEMBL6534143 0.74 GRM1 (0.42) GRM1GRM5GPR119CA1CA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082892-A2 TRIAZOLE COMPOUNDS AS ANTIBACTERIAL AGENTS AND PHARMACEUTICAL COMPOSITIONS CONTAINING THEM DR. REDDY'S LABORATORIES LTD. (IN) 2005-09-09 WO disclosed