SCHEMBL6531349

SCHEMBL6531349

COCc1nnc(-c2ccc(OC(C)C)cn2)n1-c1ccc(OC)cc1

nearest known ligand 0.48

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
OXTR P30559 10/20 0.48
AVPR1A P37288 10/20 0.48
AVPR2 P30518 2/20 0.45
L3MBTL1 Q9Y468 2/20 0.41
MEN1 O00255 1/20 0.41
KMT2A Q03164 1/20 0.41
ALDH1A1 P00352 3/20 0.40
NPSR1 Q6W5P4 3/20 0.40
POLB P06746 1/20 0.40
CRHR1 P34998 1/20 0.38
GAA P10253 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
LMNA P02545 1/20 0.38
HTT P42858 1/20 0.38
TLR8 Q9NR97 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8280980 0.89 OXTR (0.63) OXTRAVPR1AAVPR2
SCHEMBL8282035 0.71 OXTR (0.69) OXTRAVPR1AAVPR2
SCHEMBL931537 0.70 OXTR (0.68) OXTRAVPR1AAVPR2
SCHEMBL931562 0.66 OXTR (0.74) OXTRAVPR1AAVPR2
SCHEMBL6513251 0.65 OXTR (0.68) OXTRAVPR1AAVPR2
SCHEMBL12896216 0.64 MAPT (0.38)
SCHEMBL9422988 0.64 OXTR (0.58) OXTRAVPR1AAVPR2MEN1KMT2A
Hydrochloric Acid SCHEMBL10627179 0.63 OXTR (0.57) OXTRAVPR1AAVPR2MEN1KMT2A
SCHEMBL11026853 0.62 CYP1A2 (0.44) MEN1KMT2AALDH1A1HTT
SCHEMBL10624831 0.62 OXTR (0.56) OXTRAVPR1AAVPR2MEN1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005082866-A2 SUBSTITUTED 1, 2, 4- TRIAZOLE DERIVATIVES AS OXYTOCIN ANTAGONISTS PFIZER LIMITED (GB) 2005-09-09 WO disclosed