SCHEMBL6532735

SCHEMBL6532735

CC(C)(C)C(CNC(=O)O)c1nc2ccccc2[nH]1

nearest known ligand 0.51

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.50
ALOX12 P18054 1/20 0.47
CYP2C9 P11712 3/20 0.47
CYP3A4 P08684 2/20 0.47
CYP2C19 P33261 2/20 0.47
IDO1 P14902 1/20 0.47
CYP1A2 P05177 2/20 0.46
ALDH1A1 P00352 2/20 0.46
CYP2D6 P10635 1/20 0.46
FPR1 P21462 2/20 0.46
MLKL Q8NB16 1/20 0.45
POLB P06746 1/20 0.43
HTT P42858 1/20 0.43
TAAR1 Q96RJ0 1/20 0.43
BCHE P06276 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5024039 0.81 KDM4E (0.54) KMT2AALDH1A1POLB
SCHEMBL2038892 0.77 KMT2A (0.58) KMT2AALOX12CYP2C9CYP3A4CYP2C19
SCHEMBL11438595 0.75 MLKL (0.49) KMT2ACYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL11432513 0.73 KMT2A (0.45) KMT2ACYP2C9CYP3A4CYP2C19CYP1A2
SCHEMBL21247485 0.73 CNR1 (0.43) KMT2ACYP2C19CYP2D6
SCHEMBL29701262 0.72 IDO1 (0.54) KMT2AALOX12CYP2C9CYP3A4CYP2C19
SCHEMBL2937870 0.72 TSHR (0.63) KMT2AALOX12CYP2C9CYP3A4CYP2C19
SCHEMBL38663445 0.72 BCHE (0.60) KMT2AALOX12CYP2C9CYP3A4CYP2C19
SCHEMBL3842687 0.70 KMT2A (0.61) KMT2AALOX12CYP2C9CYP3A4CYP2C19
SCHEMBL36603600 0.70 KMT2A (0.61) KMT2AALOX12CYP2C9CYP3A4CYP2C19

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1286673-B8 LIGANDS OF INTEGRIN RECEPTORS ABBOTT GMBH & CO KG (DE) 2005-07-20 EP disclosed
EP-1286673-A2 LIGANDS OF INTEGRIN RECEPTORS Basf Aktiengesellschaft (DE) 2003-03-05 EP disclosed
WO-2001093840-A2 LIGANDS OF INTEGRIN RECEPTORS BASF AG (DE) 2001-12-13 WO disclosed