SCHEMBL6532743

SCHEMBL6532743

CN1CCN(c2ccc(C(=O)O)c3c2CCCC3)CC1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HTR3E A5X5Y0 1/20 0.43
HTR3B O95264 1/20 0.43
HTR3A P46098 1/20 0.43
HTR3D Q70Z44 1/20 0.43
HTR3C Q8WXA8 1/20 0.43
HTR1A P08908 2/20 0.42
HTR1D P28221 2/20 0.42
HTR1B P28222 2/20 0.42
ALDH1A1 P00352 3/20 0.41
KDM4E B2RXH2 1/20 0.41
HSD17B10 Q99714 1/20 0.41
TMEM97 Q5BJF2 1/20 0.41
SIGMAR1 Q99720 1/20 0.41
XDH P47989 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
DRD2 P14416 1/20 0.40
DRD3 P35462 1/20 0.40
HTR6 P50406 1/20 0.40
LMNA P02545 2/20 0.40
GAA P10253 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL4750860 0.81 KDM4E (0.39) ALDH1A1KDM4EHSD17B10TMEM97SIGMAR1
SCHEMBL87519 0.76 CYP1A2 (0.57) ALDH1A1KDM4EHSD17B10XDHGAA
SCHEMBL27513258 0.75 DRD2 (0.49) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL7426055 0.74 KDM4E (0.51) HTR3EHTR3BHTR3AHTR3DHTR3C
SCHEMBL11163211 0.74 KDM4E (0.47) ALDH1A1KDM4EHSD17B10DRD2DRD3
Cyclohexane SCHEMBL1538047 0.74 CYP1A2 (0.55) ALDH1A1KDM4EHSD17B10XDHGAA
SCHEMBL250454 0.74 CYP1A2 (0.55) ALDH1A1KDM4EHSD17B10XDHGAA
SCHEMBL982478 0.74 CYP1A2 (0.55) ALDH1A1KDM4EHSD17B10XDHGAA
SCHEMBL3091854 0.74 CYP1A2 (0.55) ALDH1A1KDM4EHSD17B10XDHGAA
SCHEMBL195800 0.74 CYP1A2 (0.55) ALDH1A1KDM4EHSD17B10XDHGAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005113527-A1 TETRAHYDRONAPHTHYL- PIPERAZINES AS 5-HT1B ANTAGONISTS, INVERSE AGONISTS AND PARTIAL AGONISTS PFIZER PRODUCTS INC. (US) 2005-12-01 WO disclosed