SCHEMBL6533212

SCHEMBL6533212

NC(=O)Nc1cc2cccc(C(N)=O)c2nc1-c1cccs1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PARP1 P09874 9/20 0.44
CCNE2 O96020 1/20 0.43
CDK4 P11802 1/20 0.43
CCND1 P24385 1/20 0.43
CCNE1 P24864 1/20 0.43
CDK2 P24941 1/20 0.43
IKBKB O14920 2/20 0.41
RPS6KB2 Q9UBS0 1/20 0.40
JAK2 O60674 1/20 0.40
JAK3 P52333 1/20 0.40
KDM4E B2RXH2 4/20 0.40
KMT2A Q03164 3/20 0.40
ALDH1A1 P00352 2/20 0.40
MAPT P10636 2/20 0.40
MEN1 O00255 2/20 0.40
CYP1A2 P05177 1/20 0.40
CYP3A4 P08684 1/20 0.40
CYP2D6 P10635 1/20 0.40
CYP2C19 P33261 1/20 0.40
HSD17B10 Q99714 2/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6533209 0.83 PARP1 (0.41) PARP1CCNE2CDK4CCND1CCNE1
SCHEMBL31661920 0.71 IKBKB (0.55) IKBKBRPS6KB2KDM4EKMT2AALDH1A1
SCHEMBL1385872 0.70 IKBKB (0.67) IKBKBJAK2JAK3KDM4EKMT2A
SCHEMBL7503112 0.68 KDM4E (0.40) IKBKBRPS6KB2JAK2KDM4EALDH1A1
SCHEMBL2771222 0.68 RAB9A (0.60) KDM4EKMT2AHSD17B10RAB9ASMN1; SMN2
SCHEMBL31238942 0.67 PARP1 (0.46) PARP1JAK2KDM4EKMT2AALDH1A1
SCHEMBL10406074 0.67 PARP1 (0.46) PARP1JAK2KDM4EKMT2AALDH1A1
SCHEMBL4341036 0.67 KDM4E (0.50) IKBKBRPS6KB2JAK2KDM4EKMT2A
SCHEMBL28108675 0.67 PARP1 (0.59) PARP1KDM4EALDH1A1GAA
SCHEMBL29412126 0.67 PKN1 (0.64) PARP1GAA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005105777-A1 SUBSTITUTED THIOPHENE AMIDE COMPOUNDS FOR THE TREATMENT OF INFLAMMATION PHARMACIA & UPJOHN COMPANY LLC (US) 2005-11-10 WO disclosed