SCHEMBL6533257

SCHEMBL6533257

COC(=O)C(Cc1ccc(OC(c2ccc(CC(C)C)cc2)c2cn[nH]c2)cc1)C(C)=NOCc1ccc(Cl)cc1

nearest known ligand 0.35

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 1/20 0.34
PTGS2 P35354 1/20 0.34
PPARG P37231 8/20 0.34
PPARA Q07869 8/20 0.34
MAOB P27338 1/20 0.33
CNR1 P21554 3/20 0.32
CNR2 P34972 2/20 0.32
KMT2A Q03164 1/20 0.32
AKT1 P31749 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6533825 0.94 PPARG (0.37) ROCK2PPARGPPARAAKT1
SCHEMBL6532874 0.93 PPARG (0.40) ROCK2PPARGPPARACNR1
SCHEMBL6532684 0.93 PPARG (0.38) ROCK2PPARGPPARA
SCHEMBL6533025 0.93 PPARG (0.40) PPARGPPARAMAOB
SCHEMBL6532383 0.92 PPARG (0.40) ROCK2PPARGPPARA
SCHEMBL6533886 0.89 PPARG (0.36) PPARGPPARA
SCHEMBL6532334 0.88 PPARG (0.35) PTGS2PPARGPPARA
SCHEMBL6532514 0.87 CXCR1 (0.34) PTGS2PPARGPPARA
SCHEMBL6534035 0.87 ACACB (0.38) ROCK2PPARGPPARAMAOB
SCHEMBL6533725 0.87 PPARG (0.42) PPARGPPARA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2005040127-A1 NOVEL COMPOUNDS AS AGONIST FOR PPAR GAMMA AND PPAR ALPHA, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES LTD. (KR) 2005-05-06 WO claimed
WO-2005040127-A1 NOVEL COMPOUNDS AS AGONIST FOR PPAR GAMMA AND PPAR ALPHA, METHOD FOR PREPARATION OF THE SAME, AND PHARMACEUTICAL COMPOSITION CONTAINING THE SAME LG LIFE SCIENCES LTD. (KR) 2005-05-06 WO disclosed