SCHEMBL6534368

SCHEMBL6534368

COc1ccc(-c2cc(Cl)c3ccccc3n2)cc1Cl

nearest known ligand 0.60

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ACACA Q13085 2/20 0.60
HPGD P15428 5/20 0.57
LMNA P02545 2/20 0.57
SMN1; SMN2 Q16637 2/20 0.57
KDM4E B2RXH2 5/20 0.56
ALDH1A1 P00352 4/20 0.56
HTT P42858 2/20 0.56
MAPT P10636 1/20 0.56
DHODH Q02127 3/20 0.53
KMT2A Q03164 3/20 0.52
MEN1 O00255 2/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
GAA P10253 1/20 0.50
PTGS2 P35354 1/20 0.50
NPC1 O15118 1/20 0.50
RAB9A P51151 1/20 0.50
KMO O15229 2/20 0.49
ADORA2A P29274 1/20 0.47
ADORA1 P30542 1/20 0.47
USP2 O75604 1/20 0.47

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6534192 0.89 ACACA (0.58) ACACAHPGDLMNASMN1; SMN2KDM4E
SCHEMBL6534318 0.82 MAPT (0.71) ACACAHPGDLMNASMN1; SMN2KDM4E
SCHEMBL29636789 0.82 MAPT (0.71) ACACAHPGDLMNASMN1; SMN2KDM4E
SCHEMBL6001926 0.82 ACACA (0.60) ACACAHPGDLMNASMN1; SMN2KDM4E
SCHEMBL6534274 0.82 MEN1 (0.53) ACACAHTTMAPTDHODHKMT2A
SCHEMBL6534253 0.81 TP53 (0.47) ACACAHPGDLMNASMN1; SMN2KDM4E
SCHEMBL5822925 0.81 ACACA (0.49) ACACAHPGDLMNASMN1; SMN2KDM4E
SCHEMBL9788752 0.80 DHODH (0.69) HPGDLMNASMN1; SMN2KDM4EALDH1A1
SCHEMBL3909868 0.79 HSP90AA1 (0.55) ACACAHPGDLMNASMN1; SMN2KDM4E
SCHEMBL30592743 0.78 DHODH (0.58) ACACAHPGDLMNASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1088818-B1 Quinolin-4-yl derivatives HOFFMANN LA ROCHE (CH) 2004-11-03 EP disclosed
US-6440995-B1 NMDA-RECEPTOR SUBTYPE SELECTIVE BLOCKERS HOFFMAN-LA ROCHE INC. 2002-08-27 US disclosed
EP-1088818-A1 Quinolin-4-yl derivatives F. HOFFMANN-LA ROCHE AG (CH) 2001-04-04 EP disclosed