SCHEMBL6535101

SCHEMBL6535101

CC(=O)CC(O)C=Cc1ccc(N(C)C)cc1

nearest known ligand 0.56

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
HSD17B3 P37058 1/20 0.56
APP P05067 5/20 0.46
HDAC3 O15379 2/20 0.44
HDAC4 P56524 2/20 0.44
HDAC1 Q13547 2/20 0.44
HDAC7 Q8WUI4 2/20 0.44
HDAC2 Q92769 2/20 0.44
HDAC10 Q969S8 2/20 0.44
HDAC11 Q96DB2 2/20 0.44
HDAC8 Q9BY41 2/20 0.44
HDAC6 Q9UBN7 2/20 0.44
HDAC9 Q9UKV0 2/20 0.44
HDAC5 Q9UQL6 2/20 0.44
MAOB P27338 2/20 0.43
MMP8 P22894 1/20 0.43
RELA Q04206 1/20 0.43
CRHBP P24387 1/20 0.43
CRHR2 Q13324 1/20 0.43
TLR9 Q9NR96 1/20 0.43
PTGS1 P23219 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL13306592 1.00 HSD17B3 (0.56) HSD17B3APPHDAC3HDAC4HDAC1
SCHEMBL6535451 0.76 KMT2A (0.50) APPMAOBPTGS1MAPTMAOA
SCHEMBL6535242 0.76 KMT2A (0.50) APPMAOBPTGS1MAPTMAOA
SCHEMBL24740555 0.76 APP (0.59) HSD17B3APPHDAC3HDAC4HDAC1
SCHEMBL10411806 0.76 APP (0.59) HSD17B3APPHDAC3HDAC4HDAC1
SCHEMBL10411804 0.76 APP (0.59) HSD17B3APPHDAC3HDAC4HDAC1
SCHEMBL22359184 0.74 APP (0.57) HSD17B3APPHDAC3HDAC4HDAC1
SCHEMBL9967773 0.74 APP (0.59) HSD17B3APPRELAPTGS1MAPT
SCHEMBL29332628 0.73 APP (0.44) HSD17B3APPMAOBRELAPTGS1
SCHEMBL3050207 0.72 HSD17B3 (1.00) HSD17B3APPHDAC3HDAC4HDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1038018-A4 ALDOL CONDENSATIONS BY CATALYTIC ANTIBODIES SCRIPPS RESEARCH INST (US) 2004-10-13 EP disclosed
US-6589766-B1 Use to catalyze ketone-ketone, ketone-aldehyde, aldehyde-ketone, and aldehyde-aldehyde intermolecular aldol reactions, and in some cases to catalyze their subsequent dehydration to yield aldol condensation products THE SCRIPPS RESEARCH INSTITUTE 2003-07-08 US disclosed
US-6326176-B1 ALDOL CONDENSATIONS AND CATALYTIC ANTIBODIES THE SCRIPPS RESEARCH INSTITUTE 2001-12-04 US disclosed
EP-1038018-A1 ALDOL CONDENSATIONS BY CATALYTIC ANTIBODIES The Scripps Research Institute (US) 2000-09-27 EP disclosed
WO-1999031263-A1 ALDOL CONDENSATIONS BY CATALYTIC ANTIBODIES THE SCRIPPS RESEARCH INSTITUTE (US) 1999-06-24 WO disclosed