SCHEMBL6535286

SCHEMBL6535286

COC(=O)c1ccc(Br)c(C)c1OC

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 6/20 0.41
ALDH1A1 P00352 3/20 0.41
CA1 P00915 3/20 0.41
CA2 P00918 3/20 0.41
CA9 Q16790 3/20 0.41
HPGD P15428 2/20 0.41
CA12 O43570 2/20 0.41
CA7 P43166 2/20 0.41
CA14 Q9ULX7 2/20 0.41
PDK2 Q15119 1/20 0.41
PDK4 Q16654 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
POLB P06746 3/20 0.40
LMNA P02545 1/20 0.39
TSHR P16473 1/20 0.39
HSD17B10 Q99714 4/20 0.39
GAA P10253 3/20 0.39
GLA P06280 2/20 0.39
ATM Q13315 2/20 0.39
MAPT P10636 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL977363 0.86 KDM4E (0.44) KDM4EALDH1A1CA1CA2CA9
SCHEMBL31172701 0.85 KDM4E (0.46) KDM4EALDH1A1CA1CA2CA9
SCHEMBL17041239 0.84 ALDH1A1 (0.41) KDM4EALDH1A1HPGDLMNATSHR
SCHEMBL1987207 0.84 HSD17B10 (0.51) KDM4EALDH1A1HPGDPOLBHSD17B10
SCHEMBL20146043 0.83 CA1 (0.44) KDM4EALDH1A1CA1CA2CA9
SCHEMBL17877001 0.81 CA1 (0.43) KDM4EALDH1A1CA1CA2CA9
SCHEMBL23380419 0.81 ABL1 (0.44) KDM4EALDH1A1CA1CA2CA9
SCHEMBL29825832 0.81 SOS1 (0.43) KDM4EALDH1A1CA1CA2CA9
SCHEMBL23286523 0.81 SOS1 (0.43) KDM4EALDH1A1CA1CA2CA9
SCHEMBL6852879 0.80 CA1 (0.52) KDM4EALDH1A1CA1CA2CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-3814331-B9 NOVEL LXR MODULATORS WITH BICYCLIC CORE MOIETY ORSOBIO INC (US) 2023-08-09 EP disclosed
EP-1011666-A4 ANTITHROMBOTIC AGENTS LILLY CO ELI (US) 2004-03-31 EP disclosed
EP-0997465-B1 Azaindole derivatives and their use as antithrombotic agents LILLY CO ELI (US) 2004-02-04 EP disclosed
US-6359136-B1 AZAINDOLE COMPOUND ELI LILLY AND COMPANY 2002-03-19 US disclosed
US-6265416-B1 ANTICOAGULANTS ELI LILLY AND COMPANY 2001-07-24 US disclosed
EP-1011666-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 2000-06-28 EP disclosed
WO-1998048797-A1 ANTITHROMBOTIC AGENTS ELI LILLY AND COMPANY (US) 1998-11-05 WO disclosed