SCHEMBL6852879

SCHEMBL6852879

COC(=O)c1ccc(C(=O)OC)c(OC)c1OC

nearest known ligand 0.52

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.52
CA2 P00918 3/20 0.52
CA12 O43570 2/20 0.52
CA7 P43166 2/20 0.52
CA9 Q16790 2/20 0.52
CA14 Q9ULX7 2/20 0.52
PDK2 Q15119 1/20 0.52
PDK4 Q16654 1/20 0.52
KDM4E B2RXH2 9/20 0.50
ALDH1A1 P00352 5/20 0.50
POLB P06746 3/20 0.50
HPGD P15428 3/20 0.50
TSHR P16473 2/20 0.50
LMNA P02545 1/20 0.50
NPSR1 Q6W5P4 1/20 0.50
GAA P10253 3/20 0.48
HSD17B10 Q99714 3/20 0.48
MAPT P10636 3/20 0.48
GLA P06280 2/20 0.48
ATM Q13315 2/20 0.48

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6852883 0.91 MAPT (0.52) CA1CA2CA12CA7CA9
Methyl 2,3,4-Trimethoxybenzoate SCHEMBL1434191 0.89 ALDH1A1 (0.57) KDM4EALDH1A1POLBGAAHSD17B10
SCHEMBL6240686 0.89 CA1 (0.44) CA1CA2CA12CA7CA9
SCHEMBL11046315 0.89 MAPT (0.50) CA1CA2CA12CA7CA9
SCHEMBL31172701 0.88 KDM4E (0.46) CA1CA2CA12CA7CA9
SCHEMBL11046314 0.88 CA1 (0.43) CA1CA2CA12CA7CA9
SCHEMBL3511611 0.86 TSHR (0.57) CA1CA2CA12CA7CA9
SCHEMBL18529866 0.85 ABL1 (0.49) CA1CA2CA12CA7CA9
SCHEMBL16173476 0.83 CA12 (0.52) CA1CA2CA12CA7CA9
SCHEMBL17877001 0.83 CA1 (0.43) CA1CA2CA12CA7CA9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0799827-B1 ACRYLAMIDE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME KYORIN SEIYAKU KK (JP) 2004-05-12 EP disclosed
US-5786486-A ANTIMICROBIAL, ANTITUMOR AGENTS KYORIN PHARMACEUTICAL CO., LTD. (JP) 1998-07-28 US disclosed
EP-0799827-A1 ACRYLAMIDE DERIVATIVES AND PROCESS FOR PRODUCING THE SAME KYORIN PHARMACEUTICAL CO., LTD. (JP) 1997-10-08 EP disclosed
US-4442305-A FOR USE IN CITRO OR IN VIVO THE UNITED STATES OF AMERICA AS REPRESENTED BY THE UNITED STATES DEPARTMENT OF ENERGY (US) 1984-04-10 US disclosed