SCHEMBL6535359

SCHEMBL6535359

CC(=O)CC(O)c1ccc(NC(C)=O)cc1

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
DHODH Q02127 1/20 0.54
SMN1; SMN2 Q16637 3/20 0.52
HTT P42858 1/20 0.52
L3MBTL1 Q9Y468 1/20 0.52
KMT2A Q03164 7/20 0.50
ALDH1A1 P00352 5/20 0.50
MEN1 O00255 4/20 0.50
MAPT P10636 3/20 0.50
TDP1 Q9NUW8 2/20 0.50
TSHR P16473 2/20 0.50
CA12 O43570 1/20 0.50
BRD4 O60885 1/20 0.50
NR1I2 O75469 1/20 0.50
CA1 P00915 1/20 0.50
CA2 P00918 1/20 0.50
MB P02144 1/20 0.50
CYP1A1 P04798 1/20 0.50
CA3 P07451 1/20 0.50
CYP3A4 P08684 1/20 0.50
RARG P13631 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6535180 0.85 KMT2A (0.50) SMN1; SMN2HTTKMT2AALDH1A1MEN1
SCHEMBL13306594 0.85 KMT2A (0.50) SMN1; SMN2HTTKMT2AALDH1A1MEN1
SCHEMBL6324850 0.82 DHODH (0.54) DHODHSMN1; SMN2HTTL3MBTL1KMT2A
SCHEMBL7153255 0.82 DHODH (0.54) DHODHSMN1; SMN2HTTL3MBTL1KMT2A
SCHEMBL6981790 0.81 PPID (0.51) DHODHSMN1; SMN2HTTL3MBTL1KMT2A
SCHEMBL6318456 0.81 TDP1 (0.58) DHODHSMN1; SMN2HTTL3MBTL1KMT2A
SCHEMBL9193955 0.81 DHODH (0.53) DHODHSMN1; SMN2HTTL3MBTL1KMT2A
SCHEMBL6316512 0.79 DHODH (0.51) DHODHSMN1; SMN2HTTL3MBTL1KMT2A
SCHEMBL11112670 0.79 SMN1; SMN2 (0.61) DHODHSMN1; SMN2HTTL3MBTL1KMT2A
SCHEMBL3137531 0.78 KDM4E (0.53) DHODHSMN1; SMN2HTTL3MBTL1KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1038018-A4 ALDOL CONDENSATIONS BY CATALYTIC ANTIBODIES SCRIPPS RESEARCH INST (US) 2004-10-13 EP disclosed
US-6589766-B1 Use to catalyze ketone-ketone, ketone-aldehyde, aldehyde-ketone, and aldehyde-aldehyde intermolecular aldol reactions, and in some cases to catalyze their subsequent dehydration to yield aldol condensation products THE SCRIPPS RESEARCH INSTITUTE 2003-07-08 US disclosed
US-6326176-B1 ALDOL CONDENSATIONS AND CATALYTIC ANTIBODIES THE SCRIPPS RESEARCH INSTITUTE 2001-12-04 US disclosed
EP-1038018-A1 ALDOL CONDENSATIONS BY CATALYTIC ANTIBODIES The Scripps Research Institute (US) 2000-09-27 EP disclosed
WO-1999031263-A1 ALDOL CONDENSATIONS BY CATALYTIC ANTIBODIES THE SCRIPPS RESEARCH INSTITUTE (US) 1999-06-24 WO disclosed