SCHEMBL6535646

SCHEMBL6535646

C[Si](C)(C)C#Cc1ccccc1C#Cc1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 4/20 0.50
KDM4E B2RXH2 3/20 0.50
MEN1 O00255 3/20 0.50
ALDH1A1 P00352 3/20 0.50
CYP1A2 P05177 3/20 0.50
CYP3A4 P08684 3/20 0.50
CYP2C9 P11712 3/20 0.50
HPGD P15428 3/20 0.50
CYP2C19 P33261 3/20 0.50
KMT2A Q03164 3/20 0.50
SMN1; SMN2 Q16637 3/20 0.50
MAPT P10636 3/20 0.50
HSD17B10 Q99714 2/20 0.50
APP P05067 1/20 0.50
CYP2D6 P10635 2/20 0.45
TSHR P16473 1/20 0.45
GRM5 P41594 6/20 0.44
RAB9A P51151 3/20 0.44
TP53 P04637 1/20 0.44
PKM P14618 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Diphenylacetylene SCHEMBL3842452 0.87 APP (0.60) NPC1KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL3839029 0.87 KDM4E (0.49) NPC1KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL712499 0.85 APP (0.57) NPC1KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL563613 0.84 APP (0.55) NPC1KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL2114742 0.82 APP (0.75) NPC1KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL5871989 0.82 APP (0.75) NPC1KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL5248505 0.81 APP (0.52) NPC1KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL5249596 0.81 APP (0.52) NPC1KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL23867871 0.79 APP (0.50) NPC1KDM4EMEN1ALDH1A1CYP1A2
SCHEMBL3892674 0.77 TSHR (0.46) KDM4EMEN1ALDH1A1CYP1A2CYP3A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-9676679-B2 Traceless directing groups in radical cascades: from oligoalkynes to fused helicenes without tethered initators The Florida State University Research Foundation, Inc. (US) 2017-06-13 US disclosed
US-20160145276-A1 TRACELESS DIRECTING GROUPS IN RADICAL CASCADES: FROM OLIGOALKYNES TO FUSED HELICENES WITHOUT TETHERED INITATORS The Florida State University Research Foundation, Inc 2016-05-26 US disclosed
EP-1309639-A4 COMPOSITIONS AND METHODS FOR THERMOSETTING MOLECULES IN ORGANIC COMPOSITIONS HONEYWELL INT INC (US) 2004-12-08 EP disclosed
EP-1309639-A1 COMPOSITIONS AND METHODS FOR THERMOSETTING MOLECULES IN ORGANIC COMPOSITIONS Honeywell International, Inc. (US) 2003-05-14 EP disclosed
WO-2002008308-A1 COMPOSITIONS AND METHODS FOR THERMOSETTING MOLECULES IN ORGANIC COMPOSITIONS HONEYWELL INTERNATIONAL INC. (US) 2002-01-31 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (1 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20160145276-A1 TRACELESS DIRECTING GROUPS IN RADICAL CASCADES: FROM OLIGOALKYNES TO FUSED HELICENES WITHOUT TETHERED INITATORS OR51E2, OR10J3, ORC3 NPC1 2671/4885KDM4E 3226/4885MEN1 2252/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.