SCHEMBL6535986

SCHEMBL6535986

COc1c(O)cc(-c2ccccc2)c(C=O)c1C#N

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.46
GLA P06280 2/20 0.46
MAPT P10636 2/20 0.46
LCK P06239 1/20 0.46
THRB P10828 1/20 0.46
LIMK1 P53667 1/20 0.46
LIMK2 P53671 1/20 0.46
PDE4B Q07343 3/20 0.46
PDE4A P27815 2/20 0.46
PDE4C Q08493 2/20 0.46
PDE4D Q08499 2/20 0.46
SQOR Q9Y6N5 4/20 0.44
CYP3A4 P08684 2/20 0.41
KDM4E B2RXH2 3/20 0.40
HPGD P15428 3/20 0.40
NPSR1 Q6W5P4 3/20 0.40
KMT2A Q03164 2/20 0.40
GAA P10253 2/20 0.40
PAX8 Q06710 1/20 0.40
PIM1 P11309 2/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6535860 0.80 ALDH1A1 (0.49) ALDH1A1GLAMAPTLCKTHRB
SCHEMBL6536119 0.78 ALDH1A1 (0.48) ALDH1A1GLAMAPTLCKTHRB
SCHEMBL6536102 0.76 ALDH1A1 (0.46) ALDH1A1GLAMAPTLCKTHRB
SCHEMBL6535943 0.75 ALDH1A1 (0.45) ALDH1A1GLAMAPTLCKTHRB
SCHEMBL6535983 0.70 ERN1 (0.45) ALDH1A1GLAMAPTLCKTHRB
SCHEMBL6535962 0.70 ALDH1A1 (0.40) ALDH1A1GLAMAPTLCKTHRB
SCHEMBL29672073 0.70 ERN1 (0.45) ALDH1A1GLAMAPTLCKTHRB
SCHEMBL28792537 0.69 ERN1 (0.57) ERN1
SCHEMBL29672067 0.69 ERN1 (0.57) ERN1
SCHEMBL8499935 0.69 PDE4B (0.75) ALDH1A1MAPTPDE4BPDE4APDE4C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1425015-A4 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL MYERS SQUIBB CO (US) 2004-12-15 EP disclosed
EP-1425015-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-09 EP disclosed
WO-2003015715-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-02-27 WO disclosed