SCHEMBL6535860

SCHEMBL6535860

COc1c(O)cc(-c2ccccc2)c(C=O)c1Cl

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.49
LCK P06239 1/20 0.49
GLA P06280 1/20 0.49
MAPT P10636 1/20 0.49
THRB P10828 1/20 0.49
LIMK1 P53667 1/20 0.49
LIMK2 P53671 1/20 0.49
PDE4B Q07343 4/20 0.49
PDE4A P27815 3/20 0.49
PDE4C Q08493 3/20 0.49
PDE4D Q08499 3/20 0.49
CYP3A4 P08684 1/20 0.44
ERN1 O75460 4/20 0.42
BACE1 P56817 2/20 0.42
KDM4E B2RXH2 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.40
EGFR P00533 1/20 0.40
CA1 P00915 1/20 0.40
CA2 P00918 1/20 0.40
GABRP O00591 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10973832 0.85 ALDH1A1 (0.45) ALDH1A1LCKGLAMAPTTHRB
SCHEMBL6536119 0.82 ALDH1A1 (0.48) ALDH1A1LCKGLAMAPTTHRB
SCHEMBL6535986 0.80 ALDH1A1 (0.46) ALDH1A1LCKGLAMAPTTHRB
SCHEMBL6536102 0.80 ALDH1A1 (0.46) ALDH1A1LCKGLAMAPTTHRB
SCHEMBL4276345 0.79 ALDH1A1 (0.42) ALDH1A1LCKGLAMAPTTHRB
SCHEMBL6535943 0.79 ALDH1A1 (0.45) ALDH1A1LCKGLAMAPTTHRB
SCHEMBL27625888 0.73 PDE4B (0.50) ALDH1A1MAPTPDE4BPDE4APDE4C
SCHEMBL29672073 0.73 ERN1 (0.45) ALDH1A1LCKGLAMAPTTHRB
SCHEMBL6535962 0.73 ALDH1A1 (0.40) ALDH1A1LCKGLAMAPTTHRB
SCHEMBL6535983 0.73 ERN1 (0.45) ALDH1A1LCKGLAMAPTTHRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1425015-A4 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL MYERS SQUIBB CO (US) 2004-12-15 EP disclosed
EP-1425015-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2004-06-09 EP disclosed
WO-2003015715-A2 TETRAHYDROQUINOLINE DERIVATIVES AS ANTITHROMBOTIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 2003-02-27 WO disclosed