SCHEMBL653620

SCHEMBL653620

CC(C)(C)OC(=O)N1CC[C@@H]2CN(c3cnc(Br)c(COS(C)(=O)=O)c3)C[C@@H]21

nearest known ligand 0.43

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
NR1H2 P55055 4/20 0.43
NR1H3 Q13133 2/20 0.43
RET P07949 1/20 0.39
NAMPT P43490 1/20 0.39
GPR119 Q8TDV5 11/20 0.37
CCR5 P51681 3/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL652498 0.89 RET (0.41) NR1H2NR1H3RETNAMPTGPR119
SCHEMBL3578060 0.88 CHRNB2 (0.34)
SCHEMBL652866 0.87 RET (0.42) NR1H2NR1H3RETNAMPTGPR119
SCHEMBL654453 0.84 RET (0.45) NR1H2NR1H3RETNAMPTGPR119
Hydrochloric Acid SCHEMBL653100 0.80 CHRNB2 (0.49) NR1H2NR1H3RETNAMPTGPR119
SCHEMBL652442 0.79 RET (0.50) NR1H2NR1H3RETNAMPTGPR119
SCHEMBL649860 0.79 NR1H2 (0.40) NR1H2NR1H3RETNAMPTGPR119
SCHEMBL3578532 0.77 CHRNB2 (0.38)
SCHEMBL650034 0.77 GPR119 (0.43) NR1H2NR1H3RETGPR119
SCHEMBL650737 0.77 GPR119 (0.43) NR1H2NR1H3RETGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119635-B2 Diazabicyclic central nervous system active agents ABBOTT LABORATORIES (US) 2012-02-21 US disclosed
EP-2298775-A1 Diazabicyclic central nervous system active agents Abbott Laboratories (US) 2011-03-23 EP disclosed
EP-2295437-A1 Diazabicyclic central nervous system active agents Abbott Laboratories (US) 2011-03-16 EP disclosed