SCHEMBL653688

SCHEMBL653688

CS(=O)(=O)OCC1CN(C(=O)O)CC1NCc1ccccc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
FABP6 P51161 1/20 0.40
FUCA1 P04066 1/20 0.37
GRM2 Q14416 1/20 0.37
GRM3 Q14832 1/20 0.37
HSD17B10 Q99714 2/20 0.36
ALDH1A1 P00352 2/20 0.36
MAPT P10636 1/20 0.36
HPGD P15428 1/20 0.36
NPSR1 Q6W5P4 1/20 0.36
MAOA P21397 5/20 0.35
KDM1A O60341 4/20 0.35
DRD4 P21917 1/20 0.35
EBP Q15125 1/20 0.35
DHCR7 Q9UBM7 1/20 0.35
MAOB P27338 1/20 0.35
GRIN2B Q13224 1/20 0.35
F2 P00734 1/20 0.34
PRSS1 P07477 1/20 0.34
CA1 P00915 1/20 0.34
CA2 P00918 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL652927 0.81 GRM2 (0.43) FUCA1GRM2GRM3HSD17B10NPSR1
SCHEMBL4106856 0.77 CCR5 (0.41)
SCHEMBL16053196 0.76 KDM4E (0.31) ALDH1A1TSHR
SCHEMBL28833842 0.76 CTSK (0.44) ALDH1A1TSHR
SCHEMBL23415559 0.76 CTSK (0.44) ALDH1A1TSHR
SCHEMBL3666587 0.74 FUCA1 (0.46) FUCA1GRM2GRM3HSD17B10NPSR1
SCHEMBL6102343 0.74 FUCA1 (0.46) FUCA1GRM2GRM3HSD17B10NPSR1
SCHEMBL3833535 0.74 FUCA1 (0.46) FUCA1GRM2GRM3HSD17B10NPSR1
SCHEMBL743896 0.74 FUCA1 (0.46) FUCA1GRM2GRM3HSD17B10NPSR1
SCHEMBL16656041 0.73 GRM2 (0.43) FUCA1GRM2GRM3HSD17B10NPSR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-8119635-B2 Diazabicyclic central nervous system active agents ABBOTT LABORATORIES (US) 2012-02-21 US disclosed
EP-2298775-A1 Diazabicyclic central nervous system active agents Abbott Laboratories (US) 2011-03-23 EP disclosed
EP-2295437-A1 Diazabicyclic central nervous system active agents Abbott Laboratories (US) 2011-03-16 EP disclosed